SCHEMBL16645268

SCHEMBL16645268

COC(=O)c1ccc(Nc2ncccc2N)c(F)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 4/20 0.52
HTT P42858 2/20 0.47
ALOX15 P16050 2/20 0.47
MAPT P10636 6/20 0.44
ALDH1A1 P00352 4/20 0.43
KDM4E B2RXH2 4/20 0.43
GAA P10253 2/20 0.43
HPGD P15428 2/20 0.43
GLA P06280 1/20 0.43
CASP1 P29466 1/20 0.43
CASP7 P55210 1/20 0.43
ATM Q13315 1/20 0.43
HSD17B10 Q99714 1/20 0.43
MAPK1 P28482 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.40
ROCK1 Q13464 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27451929 0.83 ALOX15 (0.45) HTTALOX15MAPTALDH1A1KDM4E
SCHEMBL6793608 0.79 CA12 (0.56) DHODHHTTALOX15MAPTALDH1A1
SCHEMBL6797385 0.79 ROCK1 (0.60) HTTALOX15MAPTALDH1A1KDM4E
SCHEMBL21311026 0.79 ROCK1 (0.48) HTTALOX15MAPTALDH1A1KDM4E
SCHEMBL27168484 0.79 ALDH1A1 (0.47) HTTALOX15MAPTALDH1A1KDM4E
SCHEMBL30777212 0.79 ALDH1A1 (0.47) HTTALOX15MAPTALDH1A1KDM4E
SCHEMBL30061686 0.79 ALDH1A1 (0.47) HTTALOX15MAPTALDH1A1KDM4E
SCHEMBL6804452 0.78 CA12 (0.48) HTTALOX15MAPTALDH1A1KDM4E
SCHEMBL31227531 0.78 CA12 (0.45) DHODHHTTALOX15MAPTALDH1A1
SCHEMBL11842891 0.77 ALDH1A1 (0.49) DHODHHTTMAPTALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015052675-A1 SUBSTITUTED DIHYDRO-BENZIMIDAZOLE COMPOUNDS AS ROR GAMMA MODULATORS GLENMARK PHARMACEUTICALS S.A. (CH) 2015-04-16 WO disclosed