SCHEMBL16645368

SCHEMBL16645368

COC(=O)c1ccc(Nc2ccncc2N)c(F)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.49
GAA P10253 3/20 0.49
KDM4E B2RXH2 3/20 0.49
GLA P06280 2/20 0.49
NUDT1 P36639 1/20 0.46
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
ROCK2 O75116 4/20 0.45
MAPT P10636 4/20 0.43
HPGD P15428 2/20 0.43
CASP1 P29466 1/20 0.43
CASP7 P55210 1/20 0.43
ATM Q13315 1/20 0.43
HSD17B10 Q99714 1/20 0.43
MAPK1 P28482 1/20 0.43
CSNK2A1 P68400 2/20 0.41
PARP1 P09874 1/20 0.41
CYP19A1 P11511 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16657402 0.79 EGFR (0.50) GAANUDT1CYP1A2CYP3A4CYP2C9
SCHEMBL16645268 0.77 DHODH (0.52) ALDH1A1GAAKDM4EGLACYP1A2
SCHEMBL16657374 0.74 ALDH1A1 (0.46) ALDH1A1GAAKDM4EGLANUDT1
SCHEMBL16345475 0.74 KDM4E (0.49) ALDH1A1GAAKDM4EGLACYP1A2
SCHEMBL3276783 0.73 MAPT (0.51) ALDH1A1GAAKDM4EGLACYP1A2
SCHEMBL31254952 0.73 MAPT (0.51) ALDH1A1GAAKDM4EGLACYP1A2
SCHEMBL1457756 0.73 KDM4E (0.61) ALDH1A1GAAKDM4EGLACYP1A2
SCHEMBL22983517 0.72 GAA (0.67) ALDH1A1GAAKDM4EROCK2MAPT
SCHEMBL22471652 0.72 CYP1A2 (0.44) ALDH1A1KDM4ENUDT1CYP1A2CYP3A4
Hydrochloric Acid SCHEMBL4418745 0.72 MAPT (0.59) ALDH1A1GAAKDM4EGLACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015052675-A1 SUBSTITUTED DIHYDRO-BENZIMIDAZOLE COMPOUNDS AS ROR GAMMA MODULATORS GLENMARK PHARMACEUTICALS S.A. (CH) 2015-04-16 WO disclosed