SCHEMBL1664862

SCHEMBL1664862

O=C(Nc1ccc(Nc2ccc(Nc3ccc(N4CCC(O)CC4)cc3)cc2)c(F)c1)c1ccc2[nH]ccc2c1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.49
RAB9A P51151 4/20 0.49
MAOA P21397 1/20 0.48
MAOB P27338 1/20 0.48
ESR1 P03372 3/20 0.44
TRPV1 Q8NER1 1/20 0.44
MAPT P10636 2/20 0.43
CHRNA7 P36544 1/20 0.42
BRAF P15056 1/20 0.42
MEN1 O00255 1/20 0.41
POLB P06746 1/20 0.41
KMT2A Q03164 1/20 0.41
MCL1 Q07820 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
EGFR P00533 1/20 0.40
F10 P00742 1/20 0.40
TNIK Q9UKE5 1/20 0.40
SMYD3 Q9H7B4 1/20 0.39
NFATC1 O95644 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1667400 0.97 NPC1 (0.51) NPC1RAB9AMAOAMAOBESR1
SCHEMBL1664865 0.97 NPC1 (0.51) NPC1RAB9AMAOAMAOBESR1
SCHEMBL1665855 0.90 MAOA (0.53) NPC1RAB9AMAOAMAOBESR1
SCHEMBL1664886 0.89 MAOB (0.58) NPC1RAB9AMAOAMAOBESR1
SCHEMBL1665857 0.89 MAOA (0.52) NPC1RAB9AMAOAMAOBESR1
SCHEMBL1664889 0.87 MAOA (0.57) NPC1RAB9AMAOAMAOBESR1
SCHEMBL1663845 0.85 ESR1 (0.47) NPC1RAB9AMAOAMAOBESR1
SCHEMBL1663842 0.85 MAOA (0.43) NPC1RAB9AMAOAMAOBESR1
SCHEMBL6120725 0.84 RAB9A (0.51) NPC1RAB9AMAPTMEN1KMT2A
SCHEMBL1664879 0.83 NPC1 (0.41) NPC1RAB9AMAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2488486-A1 HEMATOPOIETIC GROWTH FACTOR MIMETIC SMALL MOLECULE COMPOUNDS AND THEIR USES Ligand Pharmaceuticals Inc. (US) 2012-08-22 EP disclosed
WO-2011046954-A1 HEMATOPOIETIC GROWTH FACTOR MIMETIC SMALL MOLECULE COMPOUNDS AND THEIR USES LIGAND PHARMACEUTICALS INC. (US) 2011-04-21 WO disclosed