SCHEMBL16649226

SCHEMBL16649226

NC1CNCC1c1ccc(C(F)(F)F)cc1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 3/20 0.47
MAOB P27338 5/20 0.44
KDM1A O60341 4/20 0.44
KCNH2 Q12809 5/20 0.44
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
CHRNB2 P17787 2/20 0.41
CHRNA4 P43681 2/20 0.41
CHRNB4 P30926 1/20 0.41
CHRNA3 P32297 1/20 0.41
MAOA P21397 3/20 0.41
TACR1 P25103 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15055279 0.85 HTR2C (0.56) HTR2CMAOBKDM1A
SCHEMBL12813766 0.79 KDM1A (0.63) HTR2CMAOBKDM1AKCNH2CYP3A4
SCHEMBL12813765 0.79 KDM1A (0.63) HTR2CMAOBKDM1AKCNH2CYP3A4
SCHEMBL28537486 0.79 HTR2C (0.47) HTR2CMAOBKDM1AKCNH2CYP3A4
Hydrochloric Acid SCHEMBL15091771 0.77 HTR2C (0.62) HTR2CMAOBKDM1AKCNH2CYP2C19
Hydrochloric Acid SCHEMBL15091773 0.77 HTR2C (0.62) HTR2CMAOBKDM1AKCNH2CYP2C19
SCHEMBL3346427 0.76 KCNH2 (0.57) HTR2CKCNH2CYP3A4CYP2D6CYP2C9
SCHEMBL16649818 0.76 KDM1A (0.69) KDM1AKCNH2CHRNB2CHRNA4CHRNB4
SCHEMBL15729989 0.76 SLC6A3 (0.44) HTR2CMAOBKDM1A
SCHEMBL14813595 0.76 HTR2C (0.43) HTR2CMAOBKDM1AKCNH2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2681215-B1 SERINE/THREONINE KINASE INHIBITORS ARRAY BIOPHARMA INC (US) 2015-04-22 EP claimed