SCHEMBL28537486

SCHEMBL28537486

CC1CNCC1c1ccc(C(F)(F)F)cc1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 7/20 0.47
KCNH2 Q12809 5/20 0.47
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
P2RY14 Q15391 1/20 0.43
CHRNB2 P17787 2/20 0.41
CHRNA4 P43681 2/20 0.41
CHRNB4 P30926 1/20 0.41
CHRNA3 P32297 1/20 0.41
TACR1 P25103 1/20 0.40
HTR2A P28223 4/20 0.40
HTR2B P41595 4/20 0.40
AKT1 P31749 1/20 0.38
KDM1A O60341 1/20 0.38
MAOB P27338 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26516042 0.85 P2RY14 (0.56) HTR2CKCNH2P2RY14HTR2AHTR2B
SCHEMBL26114096 0.85 P2RY14 (0.56) HTR2CKCNH2P2RY14HTR2AHTR2B
SCHEMBL22958179 0.85 P2RY14 (0.56) HTR2CKCNH2P2RY14HTR2AHTR2B
SCHEMBL9776280 0.84 SLC6A2 (0.38) KCNH2CYP3A4CYP2D6CYP2C9CYP2C19
Hydrochloric Acid SCHEMBL4894281 0.83 HTR2C (0.57) HTR2CP2RY14TACR1HTR2AHTR2B
Hydrochloric Acid SCHEMBL4894283 0.83 HTR2C (0.57) HTR2CP2RY14TACR1HTR2AHTR2B
SCHEMBL12875674 0.79 HTR2C (0.55) HTR2CCHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL18848434 0.79 HTR2C (0.55) HTR2CCHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL16649226 0.79 HTR2C (0.47) HTR2CKCNH2CYP3A4CYP2D6CYP2C9
SCHEMBL14390239 0.77 HTR2C (0.43) HTR2CKCNH2CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112513021-B ROR gamma antagonist and application thereof in medicines 广东东阳光药业有限公司 2023-06-27 CN disclosed
CN-112513021-A ROR gamma antagonist and application thereof in medicine 广东东阳光药业有限公司 2021-03-16 CN disclosed