SCHEMBL16649602

SCHEMBL16649602

C[C@H](O)[C@@H](N)c1cccc(C(F)(F)F)c1F

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.47
TDO2 P48775 1/20 0.47
P2RX7 Q99572 1/20 0.42
CCR1 P32246 1/20 0.36
PDE2A O00408 3/20 0.36
MPL P40238 3/20 0.35
CTSS P25774 2/20 0.35
HDAC8 Q9BY41 1/20 0.34
EPHX2 P34913 1/20 0.34
SCN10A Q9Y5Y9 1/20 0.34
GRIN1 Q05586 1/20 0.33
GRIN2A Q12879 1/20 0.33
ACP3 P15309 1/20 0.33
SOS1 Q07889 1/20 0.33
CTSK P43235 1/20 0.33
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
HTR2B P41595 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16649567 1.00 IDO1 (0.47) IDO1TDO2P2RX7CCR1PDE2A
SCHEMBL4234796 0.82 IDO1 (0.51) IDO1TDO2P2RX7CCR1PDE2A
SCHEMBL21132890 0.82 IDO1 (0.47) IDO1TDO2P2RX7CCR1PDE2A
SCHEMBL29656429 0.82 IDO1 (0.51) IDO1TDO2P2RX7CCR1PDE2A
SCHEMBL29845425 0.82 IDO1 (0.51) IDO1TDO2P2RX7CCR1PDE2A
SCHEMBL25019477 0.82 IDO1 (0.47) IDO1TDO2P2RX7CCR1PDE2A
SCHEMBL14120782 0.82 IDO1 (0.51) IDO1TDO2P2RX7CCR1PDE2A
SCHEMBL4550765 0.82 IDO1 (0.51) IDO1TDO2P2RX7CCR1PDE2A
Hydrochloric Acid SCHEMBL25358651 0.81 IDO1 (0.54) IDO1TDO2P2RX7CCR1PDE2A
Hydrochloric Acid SCHEMBL2716131 0.81 IDO1 (0.54) IDO1TDO2P2RX7CCR1PDE2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9133187-B2 Serine/threonine kinase inhibitors ARRAY BIOPHARMA INC. (US) 2015-09-15 US claimed
EP-2681215-B1 SERINE/THREONINE KINASE INHIBITORS ARRAY BIOPHARMA INC (US) 2015-04-22 EP claimed