SCHEMBL25019477

SCHEMBL25019477

CC(O)c1cccc(C(F)(F)F)c1F

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.47
TDO2 P48775 1/20 0.47
P2RX7 Q99572 1/20 0.47
PDE2A O00408 4/20 0.40
CCR1 P32246 2/20 0.39
CTSS P25774 1/20 0.38
EPHX2 P34913 2/20 0.37
HDAC8 Q9BY41 1/20 0.37
ACP3 P15309 1/20 0.37
MPL P40238 2/20 0.36
GRIN1 Q05586 1/20 0.35
GRIN2A Q12879 1/20 0.35
SOS1 Q07889 1/20 0.35
TAS1R3 Q7RTX0 1/20 0.35
TAS1R1 Q7RTX1 1/20 0.35
TAS1R2 Q8TE23 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21132890 1.00 IDO1 (0.47) IDO1TDO2P2RX7PDE2ACCR1
SCHEMBL30991133 0.87 IDO1 (0.44) IDO1TDO2P2RX7PDE2ACCR1
SCHEMBL21132974 0.87 P2RX7 (0.39) IDO1TDO2P2RX7PDE2ASOS1
SCHEMBL25020679 0.87 P2RX7 (0.39) IDO1TDO2P2RX7PDE2ASOS1
SCHEMBL12009462 0.84 P2RX7 (0.50) IDO1TDO2P2RX7PDE2ACCR1
SCHEMBL16649602 0.82 IDO1 (0.47) IDO1TDO2P2RX7PDE2ACCR1
SCHEMBL16649567 0.82 IDO1 (0.47) IDO1TDO2P2RX7PDE2ACCR1
SCHEMBL13168657 0.82 ACP3 (0.47) P2RX7PDE2AACP3
SCHEMBL29907993 0.82 ACP3 (0.47) P2RX7PDE2AACP3
SCHEMBL29580255 0.82 ACP3 (0.47) P2RX7PDE2AACP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4219493-A1 BENZYLAMINO SUBSTITUTED PYRIDOPYRIMIDINONES AND DERIVATIVES AS SOS1 INHIBITORS Boehringer Ingelheim International GmbH (DE) 2023-08-02 EP disclosed
WO-2023022497-A1 SOS1 INHIBITOR AND USE THEREOF 주식회사 카나프테라퓨틱스 2023-02-23 WO disclosed
EP-3728254-B1 BENZYLAMINO SUBSTITUTED PYRIDOPYRIMIDINONES AND DERIVATIVES AS SOS1 INHIBITORS BOEHRINGER INGELHEIM INT (DE) 2023-02-15 EP disclosed