SCHEMBL16651

SCHEMBL16651

FC(F)(F)C=Cc1ccc(Br)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 2/20 0.42
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
HPGD P15428 1/20 0.42
RAB9A P51151 1/20 0.42
CYP2A6 P11509 1/20 0.38
MAPT P10636 3/20 0.37
MEN1 O00255 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
KMT2A Q03164 1/20 0.37
TUBB4A P04350 1/20 0.37
TUBB P07437 1/20 0.37
TUBA3C P0DPH7 1/20 0.37
TUBA1B P68363 1/20 0.37
TUBA4A P68366 1/20 0.37
TUBB4B P68371 1/20 0.37
TUBB3 Q13509 1/20 0.37
TUBB2A Q13885 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2780637 0.77 CYP2C19 (0.36) CYP2C19KDM4EALDH1A1HPGDRAB9A
SCHEMBL2780642 0.77 CYP2C19 (0.36) CYP2C19KDM4EALDH1A1HPGDRAB9A
SCHEMBL31510224 0.76 APP (0.52) CYP2C19KDM4EALDH1A1HPGDRAB9A
SCHEMBL31510225 0.76 APP (0.52) CYP2C19KDM4EALDH1A1HPGDRAB9A
SCHEMBL854913 0.76 APP (0.33)
SCHEMBL9227835 0.76 AHR (0.48) KDM4EALDH1A1CYP2A6MAPTNFE2L2
SCHEMBL9227488 0.76 NFE2L2 (0.60) CYP2C19RAB9ACYP2A6MAPTCYP3A4
SCHEMBL9227484 0.76 NFE2L2 (0.60) CYP2C19RAB9ACYP2A6MAPTCYP3A4
SCHEMBL9679616 0.76 ALDH1A1 (0.61) CYP2C19KDM4EALDH1A1HPGDRAB9A
SCHEMBL9679607 0.76 ALDH1A1 (0.61) CYP2C19KDM4EALDH1A1HPGDRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114369023-B Synthesis method and application of 2-aryl acrylate 华南理工大学 2023-01-06 CN disclosed
CN-114369023-A Synthesis method and application of 2-aryl acrylate 华南理工大学 2022-04-19 CN disclosed
CN-108658716-B Method for synthesizing olefin compound by photoinduction one-pot method 清华大学 2020-06-19 CN disclosed
CN-109651191-A A kind of difluoromethyl oxime ether derivatives and its synthetic method 华南理工大学 2019-04-19 CN disclosed
WO-2014035872-A1 TRICYCLIC ALKYNES THAT INTERACT WITH GLUCOKINASE REGULATORY PROTEIN AMGEN INC. (US) 2014-03-06 WO disclosed
WO-2013123444-A1 SULFONYL COMPOUNDS THAT INTERACT WITH GLUCOKINASE REGULATORY PROTEIN AMGEN INC. (US) 2013-08-22 WO disclosed
EP-2609081-A1 SULFONYLPIPERAZINE DERIVATIVES THAT INTERACT WITH GLUCOKINASE REGULATORY PROTEIN FOR THE TREATMENT OF DIABETES Amgen Inc. (US) 2013-07-03 EP disclosed
WO-2012027261-A1 SULFONYLPIPERAZINE DERIVATIVES THAT INTERACT WITH GLUCOKINASE REGULATORY PROTEIN FOR THE TREATMENT OF DIABETES AMGEN INC. (US) 2012-03-01 WO disclosed