SCHEMBL16655216

SCHEMBL16655216

C=C(C(=O)NO)c1ccc(CNCC23CC4CC(CC(C4)C2)C3)cc1

nearest known ligand 0.73

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 15/20 0.73
HDAC3 O15379 2/20 0.60
HDAC1 Q13547 2/20 0.60
HDAC2 Q92769 2/20 0.60
P2RX7 Q99572 2/20 0.47
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
HDAC8 Q9BY41 1/20 0.43
HDAC5 Q9UQL6 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20535185 0.84 HDAC6 (1.00) HDAC6HDAC3HDAC1HDAC2P2RX7
SCHEMBL18423583 0.78 HDAC6 (0.70) HDAC6HDAC3HDAC1HDAC2P2RX7
SCHEMBL18460736 0.78 HDAC6 (0.62) HDAC6HDAC3HDAC1HDAC2P2RX7
SCHEMBL16655138 0.77 HDAC6 (0.74) HDAC6HDAC3HDAC1HDAC2P2RX7
SCHEMBL2404317 0.75 HDAC1 (1.00) HDAC6HDAC3HDAC1HDAC2HDAC8
SCHEMBL2404324 0.75 HDAC1 (1.00) HDAC6HDAC3HDAC1HDAC2HDAC8
SCHEMBL18088397 0.72 HDAC6 (0.61) HDAC6HDAC3HDAC1HDAC2P2RX7
SCHEMBL10067533 0.72 P2RX7 (0.67) HDAC6HDAC3HDAC1HDAC2P2RX7
SCHEMBL16653762 0.71 HDAC6 (0.74) HDAC6HDAC3HDAC1HDAC2P2RX7
SCHEMBL20535184 0.71 HDAC6 (1.00) HDAC6HDAC3HDAC1HDAC2P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3062783-A1 IMAGING HISTONE DEACETYLASES WITH A RADIOTRACER USING POSITRON EMISSION TOMOGRAPHY The General Hospital Corporation DBA Massachusetts (US) 2016-09-07 EP disclosed
WO-2015058106-A1 IMAGING HISTONE DEACETYLASES WITH A RADIOTRACER USING POSITRON EMISSION TOMOGRAPHY THE GENERAL HOSPITAL CORPORATION (US) 2015-04-23 WO disclosed