SCHEMBL16655541

SCHEMBL16655541

COc1cc(B2OC(C)(C)C(C)(C)O2)cc(Cl)c1Cl

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 1/20 0.37
LPL P06858 11/20 0.35
LIPG Q9Y5X9 11/20 0.35
EGFR P00533 2/20 0.34
AAK1 Q2M2I8 1/20 0.34
SNCA P37840 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33
DGAT1 O75907 1/20 0.31
GAA P10253 1/20 0.31
NPC1 O15118 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30038611 0.84 CSF1R (0.38) CSF1RLPLLIPGEGFRAAK1
SCHEMBL529553 0.84 MEN1 (0.39) CSF1RLPLLIPGEGFRAAK1
SCHEMBL30124524 0.84 GAA (0.36) CSF1RLPLLIPGEGFRAAK1
SCHEMBL4789211 0.84 LPL (0.42) LPLLIPGEGFRCA1CA2
SCHEMBL24309439 0.83 AAK1 (0.35) LPLLIPGAAK1CA1CA2
SCHEMBL3239432 0.81 LPL (0.38) CSF1RLPLLIPGAAK1SNCA
SCHEMBL30159215 0.80 PDE4A (0.37) CSF1RLPLLIPGEGFRAAK1
SCHEMBL23797605 0.80 CSF1R (0.36) CSF1RLPLLIPGEGFRAAK1
SCHEMBL30207484 0.80 CSF1R (0.36) CSF1RLPLLIPGEGFRAAK1
SCHEMBL858457 0.80 CSF1R (0.45) CSF1RLPLLIPGEGFRAAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20210317140-A1 Heterocyclic Compounds and Methods of Use MEDIVATION TECHNOLOGIES, INC. (US) 2021-10-14 US disclosed
EP-3057970-A1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE Medivation Technologies, Inc. (US) 2016-08-24 EP disclosed
WO-2015058084-A1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE MEDIVATION TECHNOLOGIES, INC. (US) 2015-04-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210317140-A1 Heterocyclic Compounds and Methods of Use BTK, PIK3CD, PIK3CB CSF1R 2312/4885LPL 3249/4885LIPG 1740/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.