SCHEMBL16656767

SCHEMBL16656767

O=C(O)CN(CC(=O)O)[C@@H]1CCCc2ccccc21

nearest known ligand 0.58

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTT P42858 3/20 0.57
ALDH1A1 P00352 3/20 0.57
XBP1 P17861 1/20 0.57
RAB9A P51151 1/20 0.54
TRPM8 Q7Z2W7 1/20 0.49
TSHR P16473 2/20 0.48
BLM P54132 1/20 0.48
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
TAS2R14 Q9NYV8 1/20 0.45
HPGD P15428 1/20 0.45
P2RX3 P56373 2/20 0.44
P2RX2 Q9UBL9 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14463143 1.00 HTT (0.57) HTTALDH1A1XBP1RAB9ATRPM8
SCHEMBL16656814 1.00 HTT (0.57) HTTALDH1A1XBP1RAB9ATRPM8
SCHEMBL30674371 0.85 HTT (0.61) HTTALDH1A1XBP1RAB9ATRPM8
SCHEMBL13209087 0.85 HTT (0.61) HTTALDH1A1XBP1RAB9ATRPM8
SCHEMBL16656376 0.85 HTT (0.61) HTTALDH1A1XBP1RAB9ATRPM8
SCHEMBL16656359 0.85 HTT (0.61) HTTALDH1A1XBP1RAB9ATRPM8
Oxalic Acid SCHEMBL10445493 0.80 HTT (0.55) HTTALDH1A1XBP1RAB9ATRPM8
SCHEMBL12124883 0.78 HTT (0.55) HTTALDH1A1XBP1RAB9ATSHR
SCHEMBL6475089 0.77 HTT (0.49) HTTALDH1A1XBP1RAB9ATRPM8
SCHEMBL11007928 0.76 ALDH1A1 (0.48) HTTALDH1A1XBP1RAB9ATRPM8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20210009508-A1 Automated Synthesis of Small Molecules Using Chiral, Non-Racemic Boronates NATIONAL SCIENCE FOUNDATION 2021-01-14 US disclosed
US-10752577-B2 Automated synthesis of small molecules using chiral, non-racemic boronates THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 2020-08-25 US disclosed
US-20190315676-A1 AUTOMATED SYNTHESIS OF SMALL MOLECULES USING CHIRAL, NON-RACEMIC BORONATES THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS 2019-10-17 US disclosed
US-10239824-B2 Automated synthesis of small molecules using chiral, non-racemic boronates THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 2019-03-26 US disclosed
US-20170158614-A1 AUTOMATED SYNTHESIS OF SMALL MOLECULES USING CHIRAL, NON-RACEMIC BORONATES NATIONAL SCIENCE FOUNDATION 2017-06-08 US disclosed
US-9388131-B2 Automated synthesis of small molecules using chiral, non-racemic boronates THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 2016-07-12 US disclosed
US-20150329567-A1 Automated Synthesis of Small Molecules Using Chiral, Non-Racemic Boronates THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS 2015-11-19 US disclosed
US-9012658-B2 Automated synthesis of small molecules using chiral, non-racemic boronates THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 2015-04-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150329567-A1 Automated Synthesis of Small Molecules Using Chiral, Non-Racemic Boronates BTD, POLL, POLR1A HTT 4055/4885ALDH1A1 1530/4885XBP1 3112/4885
US-10752577-B2 Automated synthesis of small molecules using chiral, non-racemic boronates BTD, POLL, POLR1A HTT 4055/4885ALDH1A1 1530/4885XBP1 3112/4885
US-20170158614-A1 AUTOMATED SYNTHESIS OF SMALL MOLECULES USING CHIRAL, NON-RACEMIC BORONATES BTD, POLL, POLR1A HTT 4055/4885ALDH1A1 1530/4885XBP1 3112/4885
US-20190315676-A1 AUTOMATED SYNTHESIS OF SMALL MOLECULES USING CHIRAL, NON-RACEMIC BORONATES BTD, POLL, POLR1A HTT 4055/4885ALDH1A1 1530/4885XBP1 3112/4885
US-10239824-B2 Automated synthesis of small molecules using chiral, non-racemic boronates BTD, POLL, POLR1A HTT 4055/4885ALDH1A1 1530/4885XBP1 3112/4885
US-20210009508-A1 Automated Synthesis of Small Molecules Using Chiral, Non-Racemic Boronates BTD, POLL, POLR1A HTT 4055/4885ALDH1A1 1530/4885XBP1 3112/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.