SCHEMBL16665682

SCHEMBL16665682

C=C1/C=C\C=C/CCC(n2nc(-c3ccc(F)cc3)c3c(N)ncnc32)CC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 13/20 0.51
PIK3CD O00329 12/20 0.49
PIK3CA P42336 11/20 0.49
PIK3CB P42338 11/20 0.49
PIK3CG P48736 11/20 0.49
PRKDC P78527 11/20 0.49
ABL1 P00519 10/20 0.49
HCK P08631 10/20 0.49
SRC P12931 10/20 0.49
KDR P35968 10/20 0.49
MTOR P42345 10/20 0.49
EPHB4 P54760 10/20 0.49
PI4KB Q9UBF8 6/20 0.49
BTK Q06187 4/20 0.48
LCK P06239 1/20 0.48
LYN P07948 1/20 0.48
KDM4E B2RXH2 1/20 0.47
ALDH1A1 P00352 1/20 0.47
LMNA P02545 1/20 0.47
HTT P42858 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16665815 0.88 SRC (0.49) EGFRPIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL16665804 0.87 SRC (0.50) EGFRPIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL16665711 0.82 PIK3CD (0.62) EGFRPIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL16665783 0.80 EGFR (0.46) EGFRPIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL16665841 0.80 ATR (0.61) EGFRPIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL16665809 0.77 RET (0.43) EGFRPIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL22243265 0.75 BTK (0.67) EGFRABL1HCKSRCKDR
SCHEMBL16665849 0.75 PIK3CD (0.53) EGFRPIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL16655347 0.75 ATR (0.76) PIK3CDPIK3CAPIK3CBPIK3CGPRKDC
SCHEMBL6430687 0.74 BTK (0.82) EGFRPIK3CDPIK3CAPIK3CBPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015058084-A1 HETEROCYCLIC COMPOUNDS AND METHODS OF USE MEDIVATION TECHNOLOGIES, INC. (US) 2015-04-23 WO disclosed