SCHEMBL16666299

SCHEMBL16666299

COC(=O)C1C(=O)c2c(C)c(OC)c(C)c(C)c2OC1(C)CCC[C@@H](C)CCC[C@H](C)CCCC(C)C

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
PDE4A P27815 1/20 0.45
PDE3A Q14432 1/20 0.45
PSEN1 P49768 4/20 0.44
GSTO1 P78417 2/20 0.42
PTPN1 P18031 2/20 0.42
TTPA P49638 3/20 0.40
LMNA P02545 3/20 0.38
MAPT P10636 2/20 0.38
GSTP1 P09211 1/20 0.38
USP2 O75604 1/20 0.38
THRB P10828 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
AKT1 P31749 2/20 0.36
TRPV1 Q8NER1 1/20 0.34
NR1I2 O75469 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16671460 1.00 MEN1 (0.45) MEN1KMT2APDE4APDE3APSEN1
SCHEMBL16666298 1.00 MEN1 (0.45) MEN1KMT2APDE4APDE3APSEN1
SCHEMBL16666281 0.92 PSEN1 (0.47) MEN1KMT2APDE4APDE3APSEN1
SCHEMBL16666279 0.92 PSEN1 (0.47) MEN1KMT2APDE4APDE3APSEN1
SCHEMBL16667485 0.83 DNTT (0.41) KMT2APSEN1LMNA
SCHEMBL16667486 0.83 DNTT (0.41) KMT2APSEN1LMNA
SCHEMBL16666422 0.76 AKT1 (0.52) MEN1KMT2APDE4APDE3APSEN1
SCHEMBL16666419 0.76 AKT1 (0.52) MEN1KMT2APDE4APDE3APSEN1
SCHEMBL16666423 0.76 AKT1 (0.52) MEN1KMT2APDE4APDE3APSEN1
SCHEMBL16666352 0.74 PSEN1 (0.40) PSEN1PTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2865677-B1 Synthesis of chromane compounds and their derivatives by a copper-catalyzed conjugate addition reaction DSM IP ASSETS BV (NL) 2016-11-23 EP disclosed
WO-2015059129-A1 SYNTHESIS OF CHROMANE COMPOUNDS AND THEIR DERIVATIVES BY A COPPER-CATALYZED CONJUGATE ADDITION REACTION DSM IP ASSETS B.V. (NL) 2015-04-30 WO disclosed
EP-2865677-A1 Synthesis of chromane compounds and their derivatives by a copper-catalyzed conjugate addition reaction DSM IP Assets B.V. (NL) 2015-04-29 EP disclosed