SCHEMBL1666925

SCHEMBL1666925

CS(=O)(=O)N1CCNCC1c1c[c]ccc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 8/20 0.33
HTR2B P41595 8/20 0.33
HTR2A P28223 6/20 0.33
SMYD3 Q9H7B4 3/20 0.33
PRKD3 O94806 2/20 0.33
PRKCG P05129 2/20 0.33
PRKCB P05771 2/20 0.33
PRKCA P17252 2/20 0.33
PRKACA P17612 2/20 0.33
PRKACG P22612 2/20 0.33
PRKACB P22694 2/20 0.33
PRKCH P24723 2/20 0.33
PRKCI P41743 2/20 0.33
PRKCE Q02156 2/20 0.33
PRKCQ Q04759 2/20 0.33
PRKCZ Q05513 2/20 0.33
PRKCD Q05655 2/20 0.33
PRKD1 Q15139 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
MEN1 O00255 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12536836 0.70 PSEN1 (0.46) SMN1; SMN2MEN1CYP3A4CYP2C19KMT2A
SCHEMBL1667741 0.70 SLC18A3 (0.33) HTR2CHTR2BHTR2ATAAR1
SCHEMBL5511188 0.70 RAB9A (0.47) SMN1; SMN2MEN1CYP3A4CYP2D6CYP2C9
SCHEMBL4710814 0.70 ALDH1A1 (0.41) HTR2CHTR2BHTR2ASMYD3CYP2D6
SCHEMBL29456646 0.69 SMYD3 (0.40) HTR2CHTR2BHTR2ASMYD3SMN1; SMN2
Hydrochloric Acid SCHEMBL28210755 0.69 KMT2A (0.41) HTR2CHTR2BHTR2ASMYD3SMN1; SMN2
SCHEMBL28623338 0.68 HTR2C (0.43) HTR2CHTR2BHTR2ASMN1; SMN2MEN1
SCHEMBL7017637 0.66 HTR2C (0.38) HTR2CHTR2BHTR2APRKD3PRKCG
SCHEMBL12536865 0.65 MAPT (0.45) CYP2D6ALDH1A1LMNA
SCHEMBL28211336 0.64 ALDH1A1 (0.46) PRKD3PRKCGPRKCBPRKCAPRKACA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2488503-A1 AMINO - PYRIMIDINE COMPOUNDS AS INHIBITORS OF TBKL AND/OR IKK EPSILON Myrexis, Inc. (US) 2012-08-22 EP claimed
EP-2488503-A1 AMINO - PYRIMIDINE COMPOUNDS AS INHIBITORS OF TBKL AND/OR IKK EPSILON Myrexis, Inc. (US) 2012-08-22 EP disclosed
WO-2011046970-A1 AMINO - PYRIMIDINE COMPOUNDS AS INHIBITORS OF TBKL AND/OR IKK EPSILON MYREXIS, INC. (US) 2011-04-21 WO disclosed