SCHEMBL16670284

SCHEMBL16670284

CCOc1ccc(N(C(=O)N(C)[C@@H](C)Cc2ccccc2)S(=O)(=O)c2ccccc2C)cc1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ACACB O00763 3/20 0.46
NPY5R Q15761 2/20 0.41
MAOB P27338 1/20 0.41
RAB9A P51151 2/20 0.41
NPC1 O15118 1/20 0.41
CNR2 P34972 1/20 0.39
KMT2A Q03164 2/20 0.39
MEN1 O00255 1/20 0.39
HCRTR2 O43614 1/20 0.39
GAA P10253 1/20 0.38
MMP1 P03956 1/20 0.38
MMP13 P45452 1/20 0.38
ADAM17 P78536 1/20 0.38
TSHR P16473 1/20 0.38
MAPT P10636 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28295296 0.78 NPC1 (0.48) RAB9ANPC1KMT2AMEN1HCRTR2
SCHEMBL16681985 0.70 GAA (0.46) RAB9ANPC1CNR2KMT2AMEN1
SCHEMBL18041029 0.70 GAA (0.46) RAB9ANPC1CNR2KMT2AMEN1
SCHEMBL9179644 0.67 NPC1 (0.43) RAB9ANPC1KMT2AMMP1MMP13
SCHEMBL12204033 0.66 NPY5R (0.54) NPY5RMAOBRAB9ANPC1TSHR
Phenetole SCHEMBL8814811 0.65 LTA4H (0.49) CNR2KMT2AMEN1MAPT
SCHEMBL20943573 0.65 MAOB (0.72) MAOB
SCHEMBL20943570 0.65 MAOB (0.72) MAOB
SCHEMBL255811 0.65 ACACB (0.81) ACACBMAOB
SCHEMBL255798 0.65 ACACB (0.81) ACACBMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3060554-A1 INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION Bristol-Myers Squibb Company (US) 2016-08-31 EP disclosed
WO-2015061518-A1 INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION BRISTOL-MYERS SQUIBB COMPANY (US) 2015-04-30 WO disclosed