SCHEMBL16670528

SCHEMBL16670528

c1cnc(C2CNCCN2N2CCCCC2)cn1

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.33
ROCK2 O75116 2/20 0.32
ROCK1 Q13464 2/20 0.32
CDC42BPB Q9Y5S2 1/20 0.32
HTR2A P28223 1/20 0.32
HTR2C P28335 1/20 0.32
HTR2B P41595 1/20 0.32
CHEK1 O14757 1/20 0.31
CCNA2 P20248 1/20 0.31
CDK2 P24941 1/20 0.31
CCNA1 P78396 1/20 0.31
HRH3 Q9Y5N1 1/20 0.31
P2RX7 Q99572 1/20 0.31
KARS1 Q15046 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16670529 0.81 CHRNB2 (0.34) ALDH1A1ROCK2ROCK1CDC42BPBHRH3
SCHEMBL27978355 0.74 HTR2A (0.38) HTR2AHTR2CHTR2BP2RX7KARS1
SCHEMBL15737883 0.69 CYP3A4 (0.43) ALDH1A1HTR2CHRH3
SCHEMBL4012037 0.69 CHEK1 (0.36) ALDH1A1HTR2AHTR2CHTR2BCHEK1
SCHEMBL4020584 0.67 HRH3 (0.36) ALDH1A1ROCK2ROCK1CDC42BPBHRH3
SCHEMBL28412863 0.66 GPR119 (0.45)
SCHEMBL29757596 0.66 GPR119 (0.45)
SCHEMBL15587834 0.65 CHEK1 (0.51) CHEK1CCNA2CDK2CCNA1
SCHEMBL3460332 0.65 CHEK1 (0.51) CHEK1CCNA2CDK2CCNA1
SCHEMBL29889443 0.64 CHEK1 (0.41) CHEK1CCNA2CDK2CCNA1HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20160281165-A1 METHODS FOR DIAGNOSING, SCREENING, IDENTIFYING, MONITORING, AND TREATING ADVERSE LOCAL TISSUE REACTIONS, WHICH LEAD TO FAILURE OF ORTHOPEDIC IMPLANTS NEW YORK SOCIETY FOR THE RELIEF OF THE RUPTURED AND CRIPPLED, MAINTAINING THE HOSPITAL FOR SPECIAL SURGERY 2016-09-29 US disclosed
WO-2015061534-A1 METHODS FOR DIAGNOSING, SCREENING, IDENTIFYING, MONITORING, AND TREATING ADVERSE LOCAL TISSUE REACTIONS IN ORTHOPEDIC IMPLANTS NEW YORK SOCIETY FOR THE RUPTURED AND CRIPPLED MAINTAINING THE HOSPITAL FOR SPECIAL SURGERY (US) 2015-04-30 WO disclosed