SCHEMBL16670833

SCHEMBL16670833

O=C(Nc1cc(F)c(F)c(Cl)c1)C1CCNC1

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 3/20 0.45
KMT2A Q03164 5/20 0.42
MEN1 O00255 3/20 0.42
LMNA P02545 1/20 0.42
HPGD P15428 1/20 0.42
ALOX15 P16050 1/20 0.42
ALOX12 P18054 1/20 0.42
HTT P42858 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
MALT1 Q9UDY8 4/20 0.41
F10 P00742 1/20 0.40
ULK1 O75385 1/20 0.40
NR1I2 O75469 1/20 0.40
AHR P35869 1/20 0.40
ALDH1A1 P00352 1/20 0.39
GAA P10253 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29458465 0.90 F10 (0.46) ROCK2KMT2AMEN1LMNAALOX15
SCHEMBL22644319 0.90 F10 (0.46) ROCK2KMT2AMEN1LMNAALOX15
Hydrochloric Acid SCHEMBL22632743 0.89 F10 (0.45) ROCK2KMT2AMEN1LMNAALOX15
Hydrochloric Acid SCHEMBL16671518 0.89 F10 (0.45) ROCK2KMT2AMEN1LMNAALOX15
SCHEMBL21670326 0.84 MGLL (0.52) ROCK2KMT2AMEN1LMNAHPGD
SCHEMBL22644321 0.84 MALT1 (0.58) KMT2AMEN1LMNAHPGDALOX15
SCHEMBL18045233 0.84 F10 (0.40) ROCK2KMT2AMEN1LMNAHPGD
SCHEMBL18045234 0.84 F10 (0.40) ROCK2KMT2AMEN1LMNAHPGD
SCHEMBL29458485 0.84 MALT1 (0.58) KMT2AMEN1LMNAHPGDALOX15
Hydrochloric Acid SCHEMBL16671308 0.83 F10 (0.39) ROCK2KMT2AMEN1LMNAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3060547-A1 CARBOXAMIDE DERIVATIVES AND THE USE THEREOF AS MEDICAMENTS FOR THE TREATMENT OF HEPATITIS B Janssen Sciences Ireland UC (IE) 2016-08-31 EP disclosed
WO-2015059212-A1 CARBOXAMIDE DERIVATIVES AND THE USE THEREOF AS MEDICAMENTS FOR THE TREATMENT OF HEPATITIS B JANSSEN R&D IRELAND (IE) 2015-04-30 WO disclosed