SCHEMBL1667429

SCHEMBL1667429

CC(C)(C)N1CCC(Oc2ccc(-c3ccnc(Cl)n3)cc2C#N)CC1

nearest known ligand 0.49

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
IKBKE Q14164 17/20 0.49
TBK1 Q9UHD2 17/20 0.49
AAK1 Q2M2I8 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1667928 0.85 TBK1 (0.51) IKBKETBK1AAK1
SCHEMBL20918742 0.85 AAK1 (0.43) IKBKETBK1AAK1
SCHEMBL1669851 0.85 TBK1 (0.56) IKBKETBK1AAK1
SCHEMBL1667504 0.83 KMO (0.49) IKBKETBK1AAK1
SCHEMBL1667272 0.83 TBK1 (0.64) IKBKETBK1
SCHEMBL13467205 0.81 TBK1 (0.57) IKBKETBK1AAK1
SCHEMBL12522330 0.80 TBK1 (0.46) IKBKETBK1AAK1
SCHEMBL13280173 0.80 TBK1 (0.46) IKBKETBK1AAK1
SCHEMBL20918744 0.78 TBK1 (0.52) IKBKETBK1AAK1
SCHEMBL28408079 0.78 TBK1 (0.52) IKBKETBK1AAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2488503-A1 AMINO - PYRIMIDINE COMPOUNDS AS INHIBITORS OF TBKL AND/OR IKK EPSILON Myrexis, Inc. (US) 2012-08-22 EP disclosed
WO-2011046970-A1 AMINO - PYRIMIDINE COMPOUNDS AS INHIBITORS OF TBKL AND/OR IKK EPSILON MYREXIS, INC. (US) 2011-04-21 WO disclosed