SCHEMBL16675265

SCHEMBL16675265

[2H]C([2H])([2H])C(CC(C)(C)C)(C([2H])([2H])[2H])C([2H])([2H])C(=O)O

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.31
FFAR1 O14842 1/20 0.31
CPT2 P23786 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
HMGCR P04035 1/20 0.31
CHRM1 P11229 1/20 0.31
TBXA2R P21731 1/20 0.31
ADRA1A P35348 1/20 0.31
CYP2D6 P10635 1/20 0.30
TSHR P16473 1/20 0.30
CYP2C19 P33261 1/20 0.30
HIF1A Q16665 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16675248 0.80 KDM4E (0.46) KDM4EFFAR1CPT2TDP1HMGCR
SCHEMBL16305057 0.77 FFAR1 (0.54) KDM4EFFAR1CPT2TDP1HMGCR
SCHEMBL433760 0.69 KDM4E (0.54) KDM4EFFAR1CPT2TDP1HMGCR
SCHEMBL16675257 0.68 HMGCR (0.33) HMGCRCHRM1TBXA2RADRA1ACYP2D6
SCHEMBL17187568 0.67 KDM4E (0.52) KDM4EFFAR1CPT2TDP1HMGCR
SCHEMBL1979018 0.67 KDM4E (0.52) KDM4EFFAR1CPT2TDP1HMGCR
Methane SCHEMBL371521 0.67 KDM4E (0.52) KDM4EFFAR1CPT2TDP1HMGCR
SCHEMBL16675250 0.65 TSHR (0.35) CYP2D6TSHRCYP2C19HIF1A
Propionic Acid SCHEMBL28841722 0.64 FFAR3 (0.48) KDM4EFFAR1CPT2TDP1HMGCR
Bicarbonate SCHEMBL26105671 0.64 TSHR (0.41) KDM4EFFAR1CPT2TDP1HMGCR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9637516-B2 Betulinic acid proline derivatives as HIV inhibitors HETERO RESEARCH FOUNDATION (IN) 2017-05-02 US disclosed
US-20150337004-A1 NOVEL BETULINIC ACID PROLINE DERIVATIVES AS HIV INHIBITORS HETERO LABS LIMITED (IN) 2015-11-26 US disclosed
US-20150119373-A1 NOVEL BETULINIC ACID DERIVATIVES AS HIV INHIBITORS HETERO LABS LIMITED (IN) 2015-04-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150119373-A1 NOVEL BETULINIC ACID DERIVATIVES AS HIV INHIBITORS BET1, PGGT1B, RABGGTB KDM4E 1768/4885FFAR1 3597/4885CPT2 3312/4885
US-20150337004-A1 NOVEL BETULINIC ACID PROLINE DERIVATIVES AS HIV INHIBITORS BET1, PRR12, PELP1 KDM4E 1605/4885FFAR1 4365/4885CPT2 3708/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.