SCHEMBL1667693

SCHEMBL1667693

Cc1noc(C)c1-c1c(C(N)=O)c2cccnc2n1-c1ccc(O)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.39
HSP90AB1 P08238 1/20 0.39
BRD4 O60885 6/20 0.38
USP14 P54578 1/20 0.37
TSHR P16473 1/20 0.35
CYP3A4 P08684 3/20 0.34
CYP2C9 P11712 2/20 0.34
BRD2 P25440 2/20 0.34
BRD3 Q15059 2/20 0.34
PDE4B Q07343 2/20 0.34
CYP2C19 P33261 1/20 0.34
FTO Q9C0B1 1/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
GAA P10253 1/20 0.34
AR P10275 1/20 0.34
SLC2A1 P11166 1/20 0.34
ALDH1A1 P00352 1/20 0.33
ALOX15 P16050 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12797222 0.90 BRD4 (0.38) HSP90AA1HSP90AB1BRD4USP14TSHR
SCHEMBL1667700 0.88 BRD4 (0.36) HSP90AA1HSP90AB1BRD4USP14TSHR
SCHEMBL1667699 0.88 BRD4 (0.36) HSP90AA1HSP90AB1BRD4USP14TSHR
SCHEMBL1075535 0.84 ESR1 (0.39) BRD4TSHRCYP3A4CYP2C9BRD2
SCHEMBL30386550 0.84 ESR1 (0.39) BRD4TSHRCYP3A4CYP2C9BRD2
SCHEMBL1667702 0.84 BRD4 (0.36) BRD4USP14TSHRCYP3A4CYP2C9
SCHEMBL1668109 0.80 BRD4 (0.38) BRD4USP14TSHRCYP3A4CYP2C9
SCHEMBL1667668 0.80 HSP90AA1 (0.39) HSP90AA1HSP90AB1USP14CYP2C9CYP2C19
SCHEMBL1667681 0.79 BRD4 (0.37) BRD4TSHRCYP3A4CYP2C9CYP2C19
SCHEMBL1667684 0.79 BRD4 (0.37) BRD4TSHRCYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011042474-A1 NOVEL ESTROGEN RECEPTOR LIGANDS KARO BIO AB (SE) 2011-04-14 WO claimed
WO-2011042474-A1 NOVEL ESTROGEN RECEPTOR LIGANDS KARO BIO AB (SE) 2011-04-14 WO disclosed
WO-2011042474-A1 NOVEL ESTROGEN RECEPTOR LIGANDS KARO BIO AB (SE) 2011-04-14 WO disclosed