SCHEMBL1667702

SCHEMBL1667702

Cc1noc(C)c1-c1c(C(=N)NO)c2cccnc2n1-c1ccc(O)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 6/20 0.36
CYP1A2 P05177 9/20 0.34
CYP3A4 P08684 8/20 0.34
CYP2C19 P33261 7/20 0.34
ALOX15 P16050 7/20 0.34
CLK4 Q9HAZ1 6/20 0.34
HSD17B10 Q99714 5/20 0.34
USP2 O75604 5/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2D6 P10635 4/20 0.33
MEN1 O00255 3/20 0.33
LMNA P02545 3/20 0.33
KMT2A Q03164 3/20 0.33
MAPT P10636 2/20 0.33
TDP1 Q9NUW8 2/20 0.33
KDM4E B2RXH2 1/20 0.33
HPGD P15428 1/20 0.33
ALDH1A1 P00352 5/20 0.33
USP14 P54578 1/20 0.33
TSHR P16473 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12797222 0.88 BRD4 (0.38) BRD4CYP1A2CYP3A4CYP2C19ALOX15
SCHEMBL1670152 0.85 FTO (0.35) BRD4CYP1A2CYP3A4CYP2C19ALOX15
SCHEMBL1077681 0.85 ESR1 (0.38) BRD4CYP1A2CYP3A4CYP2C19ALOX15
SCHEMBL1670092 0.84 ESR1 (0.34) BRD4CYP1A2CYP3A4CYP2C19ALOX15
SCHEMBL1667693 0.84 HSP90AA1 (0.39) BRD4CYP1A2CYP3A4CYP2C19ALOX15
SCHEMBL1076152 0.83 CYP1A2 (0.35) BRD4CYP1A2CYP3A4CYP2C19ALOX15
SCHEMBL1667589 0.83 BRD4 (0.33) BRD4CYP1A2CYP3A4CYP2C19ALOX15
SCHEMBL1670139 0.83 USP14 (0.32) USP14
SCHEMBL1667699 0.82 BRD4 (0.36) BRD4CYP1A2CYP3A4CYP2C19ALOX15
SCHEMBL1667700 0.82 BRD4 (0.36) BRD4CYP1A2CYP3A4CYP2C19ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011042474-A1 NOVEL ESTROGEN RECEPTOR LIGANDS KARO BIO AB (SE) 2011-04-14 WO claimed
WO-2011042474-A1 NOVEL ESTROGEN RECEPTOR LIGANDS KARO BIO AB (SE) 2011-04-14 WO disclosed