SCHEMBL16684841

SCHEMBL16684841

CC1(C)CCc2ccc(N3CCC(C(N)=O)C3)cc2O1

nearest known ligand 0.40

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 3/20 0.40
NOTUM Q6P988 8/20 0.39
PDK2 Q15119 1/20 0.39
ALDH1A1 P00352 1/20 0.37
MAPT P10636 1/20 0.37
RORC P51449 1/20 0.36
PRKDC P78527 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16695101 1.00 IRAK4 (0.40) IRAK4NOTUMPDK2ALDH1A1MAPT
SCHEMBL16695084 0.91 GHSR (0.41) IRAK4NOTUMPDK2ALDH1A1MAPT
SCHEMBL16695566 0.90 NOTUM (0.51) NOTUM
SCHEMBL21340137 0.87 MAPT (0.43) NOTUMPDK2ALDH1A1MAPT
SCHEMBL16695388 0.81 NOTUM (0.51) NOTUM
SCHEMBL16684690 0.74 NOTUM (0.47) NOTUMPDK2
SCHEMBL16695100 0.74 NOTUM (0.47) NOTUMPDK2
SCHEMBL16695146 0.74 NOTUM (0.47) NOTUMPDK2
SCHEMBL16695065 0.73 NOTUM (0.43) NOTUMPDK2RORC
SCHEMBL16695078 0.73 NOTUM (0.43) NOTUMPDK2RORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3063141-A1 N-(1-HYDROXY-3-(PYRROLIDINYL)PROPAN-2-YL)PYRROLIDINE-3-CARBOXAMIDE DERIVATIVES AS GLUCOSYLCERAMIDE SYNTHASE INHIBITORS BioMarin Pharmaceutical Inc. (US) 2016-09-07 EP disclosed
WO-2015065937-A1 N-(1-HYDROXY-3-(PYRROLIDINYL)PROPAN-2-YL)PYRROLIDINE-3-CARBOXAMIDE DERIVATIVES AS GLUCOSYLCERAMIDE SYNTHASE INHIBITORS BIOMARIN PHARMACEUTICAL INC. (US) 2015-05-07 WO disclosed
WO-2015065937-A1 N-(1-HYDROXY-3-(PYRROLIDINYL)PROPAN-2-YL)PYRROLIDINE-3-CARBOXAMIDE DERIVATIVES AS GLUCOSYLCERAMIDE SYNTHASE INHIBITORS BIOMARIN PHARMACEUTICAL INC. (US) 2015-05-07 WO disclosed