SCHEMBL1669154

SCHEMBL1669154

COC(=O)Cc1ccc(O)c(C2(c3ccccc3)CCN(C(=O)OC(C)(C)C)CC2)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRD1 P41143 2/20 0.51
OPRK1 P41145 1/20 0.51
TSHR P16473 2/20 0.47
ALOX15 P16050 1/20 0.47
ATM Q13315 1/20 0.47
TACR1 P25103 1/20 0.46
JAK2 O60674 1/20 0.44
JAK1 P23458 1/20 0.44
ALDH1A1 P00352 1/20 0.43
GAA P10253 1/20 0.43
GFER P55789 1/20 0.43
HDAC1 Q13547 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
PDK2 Q15119 1/20 0.41
GPR119 Q8TDV5 2/20 0.40
STS P08842 1/20 0.40
ANO1 Q5XXA6 1/20 0.40
ACHE P22303 1/20 0.39
KDM4E B2RXH2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16511858 0.90 OPRD1 (0.48) OPRD1OPRK1TSHRALOX15ATM
SCHEMBL1668912 0.87 OPRD1 (0.51) OPRD1OPRK1TSHRALOX15ATM
SCHEMBL16499539 0.86 OPRD1 (0.52) OPRD1OPRK1TSHRALOX15ATM
SCHEMBL16498943 0.85 OPRD1 (0.52) OPRD1OPRK1TSHRALOX15ATM
SCHEMBL16498945 0.85 OPRD1 (0.52) OPRD1OPRK1TSHRALOX15ATM
SCHEMBL1668509 0.85 JAK2 (0.45) TSHRALOX15ATMTACR1JAK2
SCHEMBL1669123 0.84 OPRD1 (0.51) OPRD1OPRK1TSHRALOX15ATM
SCHEMBL16499347 0.83 OPRD1 (0.50) OPRD1OPRK1TSHRALOX15ATM
SCHEMBL1668586 0.83 OPRD1 (0.48) OPRD1OPRK1TSHRALOX15ATM
SCHEMBL12801231 0.82 OPRD1 (0.47) OPRD1OPRK1TSHRALOX15ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011048409-A1 CYCLIC AMINE DERIVATIVES HAVING BETA2 ADRENERGIC RECEPTOR AGONIST AND MUSCARINIC RECEPTOR ANTAGONIST ACTIVITY ASTRAZENECA AB (SE) 2011-04-28 WO disclosed
WO-2011048409-A1 CYCLIC AMINE DERIVATIVES HAVING BETA2 ADRENERGIC RECEPTOR AGONIST AND MUSCARINIC RECEPTOR ANTAGONIST ACTIVITY ASTRAZENECA AB (SE) 2011-04-28 WO disclosed