SCHEMBL16693133

SCHEMBL16693133

Cc1csc2cc(/C=N/O)ccc12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.42
KDM4E B2RXH2 4/20 0.40
ALDH1A1 P00352 4/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
HTT P42858 2/20 0.36
PTGS1 P23219 1/20 0.36
PTGS2 P35354 1/20 0.36
POLB P06746 1/20 0.36
PKM P14618 1/20 0.36
KMT2A Q03164 5/20 0.35
MEN1 O00255 3/20 0.35
LMNA P02545 1/20 0.35
MAPT P10636 1/20 0.35
ALOX12 P18054 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
GAA P10253 3/20 0.35
MAPK1 P28482 2/20 0.35
ACHE P22303 1/20 0.33
GFER P55789 1/20 0.33
NPC1 O15118 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16693082 1.00 CYP2A6 (0.42) CYP2A6KDM4EALDH1A1L3MBTL1HTT
SCHEMBL16693175 0.88 CYP2A6 (0.51) CYP2A6KDM4EALDH1A1L3MBTL1HTT
SCHEMBL16687131 0.80 ALDH1A1 (0.40) KDM4EALDH1A1L3MBTL1HTTPOLB
SCHEMBL16687130 0.80 ALDH1A1 (0.40) KDM4EALDH1A1L3MBTL1HTTPOLB
SCHEMBL16693174 0.77 CYP2A6 (0.42) CYP2A6ALDH1A1PTGS1PTGS2PKM
SCHEMBL16693081 0.77 CYP2A6 (0.42) CYP2A6KDM4EALDH1A1PTGS1PTGS2
SCHEMBL16693190 0.76 KDM4E (0.37) KDM4EALDH1A1L3MBTL1HTTPOLB
SCHEMBL424317 0.70 CYP2A6 (0.48) CYP2A6KDM4EALDH1A1LMNAMAPT
SCHEMBL2166114 0.70 ALDH1A1 (0.50) KDM4EALDH1A1L3MBTL1HTTPOLB
SCHEMBL1937076 0.70 ALDH1A1 (0.50) KDM4EALDH1A1L3MBTL1HTTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015066371-A1 SPIRO-OXADIAZOLINE COMPOUNDS AS AGONISTS OF α-7-NICOTINIC ACETYLCHOLINE RECEPTORS FORUM PHARMACEUTICALS, INC. (US) 2015-05-07 WO disclosed