SCHEMBL16693174

SCHEMBL16693174

C=Cc1ccc2c(C)csc2c1

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.42
TP53 P04637 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
ALDH1A1 P00352 2/20 0.36
ESR1 P03372 1/20 0.34
ESR2 Q92731 1/20 0.34
TRPA1 O75762 1/20 0.33
MAPT P10636 1/20 0.33
PKM P14618 1/20 0.33
PTGS1 P23219 1/20 0.33
PTGS2 P35354 1/20 0.33
CHRNA7 P36544 1/20 0.32
HTR3A P46098 1/20 0.32
LRRK2 Q5S007 1/20 0.31
CYP17A1 P05093 1/20 0.30
LMNA P02545 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14341667 0.85 CYP2A6 (0.55) CYP2A6TP53TDP1ALDH1A1ESR1
SCHEMBL16693081 0.81 CYP2A6 (0.42) CYP2A6TDP1ALDH1A1MAPTPTGS1
SCHEMBL16693082 0.77 CYP2A6 (0.42) CYP2A6ALDH1A1MAPTPKMPTGS1
SCHEMBL16693133 0.77 CYP2A6 (0.42) CYP2A6ALDH1A1MAPTPKMPTGS1
SCHEMBL4420015 0.75 CYP2A6 (0.58) CYP2A6ALDH1A1MAPTPTGS1PTGS2
SCHEMBL424317 0.74 CYP2A6 (0.48) CYP2A6TP53TDP1ALDH1A1MAPT
SCHEMBL28073641 0.72 PKM (0.39) TP53TDP1ALDH1A1MAPTPKM
SCHEMBL13950998 0.71 CYP2A6 (0.46) CYP2A6ALDH1A1MAPTCHRNA7HTR3A
SCHEMBL2095399 0.71 CYP2A6 (0.46) CYP2A6TP53TDP1ALDH1A1MAPT
SCHEMBL2092747 0.71 CYP2A6 (0.71) CYP2A6TP53MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015066371-A1 SPIRO-OXADIAZOLINE COMPOUNDS AS AGONISTS OF α-7-NICOTINIC ACETYLCHOLINE RECEPTORS FORUM PHARMACEUTICALS, INC. (US) 2015-05-07 WO disclosed