SCHEMBL16693166

SCHEMBL16693166

CCOC(=O)c1cc2cc(F)cc(F)c2o1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR35 Q9HC97 1/20 0.45
HDAC4 P56524 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
TSHR P16473 1/20 0.42
AKR1B1 P15121 1/20 0.41
MAOB P27338 3/20 0.40
TRPM8 Q7Z2W7 1/20 0.40
PTPN11 Q06124 1/20 0.39
KDM4E B2RXH2 3/20 0.39
ALDH1A1 P00352 2/20 0.39
MAPT P10636 1/20 0.39
CASP1 P29466 1/20 0.39
CASP7 P55210 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39
HPGD P15428 1/20 0.39
CYP2C19 P33261 1/20 0.39
MAOA P21397 1/20 0.38
GAA P10253 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16046551 0.88 GPR35 (0.45) GPR35HDAC4HDAC6TSHRAKR1B1
SCHEMBL13725141 0.87 PIM1 (0.45) GPR35HDAC4HDAC6AKR1B1MAOB
SCHEMBL931539 0.85 MAOB (0.51) GPR35HDAC4HDAC6TSHRAKR1B1
SCHEMBL29540395 0.83 GPR35 (0.60) GPR35HDAC4HDAC6AKR1B1MAOB
SCHEMBL19744146 0.83 GPR35 (0.60) GPR35HDAC4HDAC6AKR1B1MAOB
SCHEMBL20559444 0.83 MAPT (0.44) GPR35PTPN11KDM4EALDH1A1MAPT
SCHEMBL19188041 0.83 DHODH (0.41) GPR35HDAC4HDAC6AKR1B1MAOB
SCHEMBL2303899 0.82 MAOA (0.51) HDAC4HDAC6TSHRMAOBKDM4E
SCHEMBL16684605 0.78 MAOB (0.51) TSHRAKR1B1MAOBKDM4EALDH1A1
SCHEMBL26244513 0.77 AKR1B1 (0.42) HDAC4HDAC6AKR1B1MAOBKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015066371-A1 SPIRO-OXADIAZOLINE COMPOUNDS AS AGONISTS OF α-7-NICOTINIC ACETYLCHOLINE RECEPTORS FORUM PHARMACEUTICALS, INC. (US) 2015-05-07 WO disclosed