SCHEMBL1670092

SCHEMBL1670092

Cc1noc(C)c1-c1c(C(=N)NO)c2ncccc2n1-c1ccc(O)cc1

nearest known ligand 0.34

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 2/20 0.34
ESR2 Q92731 2/20 0.34
USP14 P54578 4/20 0.33
BRD4 O60885 6/20 0.32
ALDH1A1 P00352 2/20 0.30
ALOX15 P16050 2/20 0.30
L3MBTL1 Q9Y468 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2D6 P10635 1/20 0.30
TSHR P16473 1/20 0.30
CYP2C19 P33261 1/20 0.30
HSD17B10 Q99714 1/20 0.30
CLK4 Q9HAZ1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1077681 0.85 ESR1 (0.38) ESR1ESR2BRD4ALDH1A1ALOX15
SCHEMBL1667702 0.84 BRD4 (0.36) ESR1ESR2USP14BRD4ALDH1A1
SCHEMBL1670089 0.82 ESR1 (0.34) ESR1ESR2USP14BRD4
SCHEMBL1670091 0.82 ESR1 (0.34) ESR1ESR2USP14BRD4
SCHEMBL2311175 0.82 BRD4 (0.34) ESR1ESR2USP14BRD4ALDH1A1
SCHEMBL1667689 0.80 BRD4 (0.34) ESR1ESR2USP14BRD4ALOX15
SCHEMBL1670810 0.79 BRD4 (0.34) ESR1ESR2BRD4ALOX15CYP1A2
SCHEMBL1076152 0.78 CYP1A2 (0.35) ESR1USP14BRD4ALDH1A1ALOX15
SCHEMBL1077416 0.78 PTGDR2 (0.39) BRD4ALDH1A1ALOX15CYP1A2CYP3A4
SCHEMBL1078053 0.78 PIK3CD (0.36) BRD4ALDH1A1ALOX15CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011042474-A1 NOVEL ESTROGEN RECEPTOR LIGANDS KARO BIO AB (SE) 2011-04-14 WO claimed