SCHEMBL1670091

SCHEMBL1670091

Cc1noc(C)c1-c1c(C(N)=NO)c2ncccc2n1-c1ccc(O)cc1

nearest known ligand 0.34

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 2/20 0.34
ESR2 Q92731 2/20 0.34
USP14 P54578 4/20 0.33
BRD4 O60885 5/20 0.32
ADORA3 P0DMS8 3/20 0.32
CHEK1 O14757 1/20 0.30
NTRK1 P04629 1/20 0.30
PIM1 P11309 1/20 0.30
CDK2 P24941 1/20 0.30
CSNK2A1 P68400 1/20 0.30
REN P00797 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1670089 1.00 ESR1 (0.34) ESR1ESR2USP14BRD4ADORA3
SCHEMBL1077417 0.85 ESR1 (0.38) ESR1ESR2BRD4
SCHEMBL1077420 0.85 ESR1 (0.38) ESR1ESR2BRD4
SCHEMBL1667700 0.84 BRD4 (0.36) ESR1ESR2USP14BRD4ADORA3
SCHEMBL1667699 0.84 BRD4 (0.36) ESR1ESR2USP14BRD4ADORA3
SCHEMBL1670092 0.82 ESR1 (0.34) ESR1ESR2USP14BRD4
SCHEMBL2311182 0.82 BRD4 (0.34) ESR1ESR2USP14BRD4
SCHEMBL2313824 0.82 BRD4 (0.34) ESR1ESR2USP14BRD4
SCHEMBL1667683 0.80 BRD4 (0.34) ESR1ESR2USP14BRD4
SCHEMBL1667686 0.80 BRD4 (0.34) ESR1ESR2USP14BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011042474-A1 NOVEL ESTROGEN RECEPTOR LIGANDS KARO BIO AB (SE) 2011-04-14 WO claimed