SCHEMBL16701366

SCHEMBL16701366

Nc1nc(Cl)cc(N2CCN(C(=O)O)CC2)n1

nearest known ligand 0.63

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.59
CYP1A2 P05177 1/20 0.59
CYP2D6 P10635 1/20 0.59
LMNA P02545 2/20 0.56
KMT2A Q03164 1/20 0.55
HRH4 Q9H3N8 5/20 0.43
HRH3 Q9Y5N1 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.41
S1PR2 O95136 1/20 0.41
ALOX12 P18054 1/20 0.41
HTT P42858 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
GFER P55789 1/20 0.40
HTR3A P46098 1/20 0.40
CRHBP P24387 1/20 0.40
CRHR2 Q13324 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1774435 0.94 MAPT (0.54) MAPTCYP1A2CYP2D6LMNAKMT2A
SCHEMBL18153268 0.84 HRH4 (0.41) MAPTCYP1A2CYP2D6LMNAKMT2A
SCHEMBL11963431 0.82 GBA1 (0.42) MAPTCYP1A2CYP2D6LMNAKMT2A
SCHEMBL3779757 0.80 LMNA (0.55) MAPTCYP1A2CYP2D6LMNAKMT2A
SCHEMBL1579732 0.79 GAA (0.40) MAPTCYP1A2CYP2D6LMNAHTT
SCHEMBL1318180 0.79 MAPT (0.72) MAPTCYP1A2CYP2D6LMNAKMT2A
SCHEMBL3719291 0.79 MAPT (0.72) MAPTCYP1A2CYP2D6LMNAKMT2A
SCHEMBL18153411 0.78 GBA1 (0.54)
SCHEMBL21796761 0.78 LMNA (0.44) MAPTCYP1A2LMNAHRH4
SCHEMBL27908906 0.78 KMT2A (0.62) MAPTCYP1A2CYP2D6LMNAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015069752-A9 ACETYLCHOLINE BINDING PROTEIN LIGANDS, COOPERATIVE NACHR MODULATORS AND METHODS FOR MAKING AND USING THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2015-07-09 WO disclosed
WO-2015069752-A1 ACETYLCHOLINE BINDING PROTEIN LIGANDS, COOPERATIVE NACHR MODULATORS AND METHODS FOR MAKING AND USING THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2015-05-14 WO disclosed