SCHEMBL16704292

SCHEMBL16704292

CCC/N=C/c1ccc2c(c1)OCO2

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.58
KDM4E B2RXH2 2/20 0.58
ALOX15 P16050 1/20 0.58
DYRK3 O43781 2/20 0.52
PIM1 P11309 2/20 0.52
CDK5 Q00535 2/20 0.52
DYRK1A Q13627 2/20 0.52
CDK5R1 Q15078 2/20 0.52
DYRK2 Q92630 2/20 0.52
DYRK1B Q9Y463 2/20 0.52
CSNK2A2 P19784 1/20 0.52
CSNK2B P67870 1/20 0.52
CSNK2A1 P68400 1/20 0.52
CSNK2A3 Q8NEV1 1/20 0.52
CYP3A4 P08684 3/20 0.51
ATM Q13315 1/20 0.51
GSK3A P49840 2/20 0.51
GSK3B P49841 2/20 0.51
MAPT P10636 3/20 0.50
KMT2A Q03164 3/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3031855 1.00 ALDH1A1 (0.58) ALDH1A1KDM4EALOX15DYRK3PIM1
SCHEMBL4454930 0.91 ALDH1A1 (0.62) ALDH1A1KDM4EALOX15DYRK3PIM1
SCHEMBL4454927 0.91 ALDH1A1 (0.62) ALDH1A1KDM4EALOX15DYRK3PIM1
SCHEMBL4449592 0.87 CYP3A4 (0.54) ALDH1A1KDM4EALOX15DYRK3PIM1
SCHEMBL4449591 0.87 CYP3A4 (0.54) ALDH1A1KDM4EALOX15DYRK3PIM1
SCHEMBL16168568 0.81 ALDH1A1 (0.55) ALDH1A1KDM4EALOX15CYP3A4ATM
SCHEMBL5452087 0.81 ALDH1A1 (0.62) ALDH1A1KDM4EALOX15CYP3A4ATM
SCHEMBL14627221 0.81 ALDH1A1 (0.62) ALDH1A1KDM4EALOX15CYP3A4ATM
SCHEMBL11558188 0.81 ALDH1A1 (0.58) ALDH1A1KDM4EALOX15CYP3A4ATM
SCHEMBL11558191 0.81 ALDH1A1 (0.58) ALDH1A1KDM4EALOX15CYP3A4ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015069766-A1 DUPA-INDENOISOQUINOLINE CONJUGATES PURDUE RESEARCH FOUNDATION (US) 2015-05-14 WO disclosed