SCHEMBL16705333

SCHEMBL16705333

C[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)c1cccc2ccccc12)C(=O)ON

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.56
CTSB P07858 3/20 0.54
CTSV O60911 1/20 0.54
CTSL P07711 1/20 0.54
CTSS P25774 1/20 0.54
CAPN1 P07384 1/20 0.52
ELANE P08246 4/20 0.48
KDM4E B2RXH2 2/20 0.46
ALDH1A1 P00352 2/20 0.46
TACR3 P29371 1/20 0.46
PKM P14618 1/20 0.46
PSMB5 P28074 4/20 0.46
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
HPGD P15428 1/20 0.44
KCNA5 P22460 1/20 0.44
KLKB1 P03952 1/20 0.43
F10 P00742 1/20 0.43
GPR139 Q6DWJ6 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12518059 0.88 BACE1 (0.61) BACE1CTSBCTSVCTSLCTSS
SCHEMBL12463981 0.82 MMP9 (0.60) BACE1CTSBCTSVCTSLCTSS
SCHEMBL16571252 0.80 BACE1 (0.62) BACE1CTSBCTSVCTSLCTSS
SCHEMBL8017638 0.80 CCR3 (0.58) BACE1CTSBCTSVCTSLCTSS
SCHEMBL8010564 0.79 CCR3 (0.62) BACE1CTSBCTSVCTSLCTSS
SCHEMBL9716712 0.79 ELANE (0.64) BACE1CTSBCTSVCTSLCTSS
SCHEMBL10658026 0.79 ELANE (0.64) BACE1CTSBCTSVCTSLCTSS
SCHEMBL9830992 0.79 MEN1 (0.58) BACE1CTSBCTSVCTSLCTSS
SCHEMBL9830982 0.79 MEN1 (0.58) BACE1CTSBCTSVCTSLCTSS
SCHEMBL8008852 0.79 CCR3 (0.55) BACE1CTSBCTSVCTSLCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2526116-B1 PYRUVAMIDE COMPOUNDS AS INHIBITORS OF DUST MITE GROUP 1 PEPTIDASE ALLERGEN ST GEORGES HOSP MEDICAL SCHOOL (GB) 2015-05-13 EP disclosed