SCHEMBL1670722

SCHEMBL1670722

OB(O)c1ccc(C(F)(F)F)cc1C(F)(F)F.OB(O)c1ccc(F)cc1F

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.40
POLQ O75417 2/20 0.39
MGLL Q99685 2/20 0.38
PDE2A O00408 2/20 0.37
CYP1A1 P04798 1/20 0.37
CYP1B1 Q16678 1/20 0.37
LIPE Q05469 2/20 0.36
ORAI1 Q96D31 1/20 0.34
ORAI2 Q96SN7 1/20 0.34
ORAI3 Q9BRQ5 1/20 0.34
TRPV6 Q9H1D0 1/20 0.34
SCN8A Q9UQD0 1/20 0.33
SCN10A Q9Y5Y9 1/20 0.33
MTOR P42345 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29349652 0.87 CES2 (0.50) CES2POLQMGLLPDE2AORAI1
SCHEMBL496773 0.87 CES2 (0.50) CES2POLQMGLLPDE2AORAI1
SCHEMBL29755537 0.83 PDE2A (0.50) CES2MGLLPDE2AORAI1ORAI2
SCHEMBL536190 0.83 IDO1 (0.42) MGLLLIPEORAI1ORAI2ORAI3
SCHEMBL582110 0.83 PDE2A (0.50) CES2MGLLPDE2AORAI1ORAI2
SCHEMBL29825643 0.83 IDO1 (0.42) MGLLLIPEORAI1ORAI2ORAI3
SCHEMBL1670723 0.81 CES2 (0.36) CES2POLQMGLLPDE2ACYP1A1
SCHEMBL39406 0.79 CES2 (0.43) CES2ORAI1ORAI2ORAI3TRPV6
SCHEMBL29395656 0.79 CES2 (0.43) CES2ORAI1ORAI2ORAI3TRPV6
SCHEMBL1668958 0.79 MGLL (0.42) CES2POLQMGLLPDE2AORAI1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2485678-A1 COFERONS AND METHODS OF MAKING AND USING THEM Cornell University (US) 2012-08-15 EP disclosed
WO-2011043817-A1 COFERONS AND METHODS OF MAKING AND USING THEM CORNELL UNIVERSITY (US) 2011-04-14 WO disclosed