SCHEMBL1670917

SCHEMBL1670917

Cc1noc(C)c1-n1c(C=O)c(C)c(Br)c1-c1ccc(O)cc1F

nearest known ligand 0.38

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TTR P02766 1/20 0.38
ERN1 O75460 3/20 0.35
ESR1 P03372 11/20 0.33
HSP90AB1 P08238 1/20 0.32
HTT P42858 1/20 0.31
ESR2 Q92731 5/20 0.31
NSD3 Q9BZ95 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12801005 0.90 TTR (0.34) TTRESR1HSP90AB1ESR2NSD3
SCHEMBL1670320 0.89 ESR1 (0.34) TTRESR1HSP90AB1ESR2
SCHEMBL1670615 0.89 ESR1 (0.34) TTRESR1HSP90AB1ESR2
SCHEMBL1671741 0.86 ERN1 (0.35) TTRERN1
SCHEMBL1671021 0.78 ESR1 (0.34) ESR1HSP90AB1ESR2
SCHEMBL1671020 0.78 ESR1 (0.34) ESR1HSP90AB1ESR2
SCHEMBL1670649 0.72 ESR1 (0.35) TTRESR1HSP90AB1ESR2
SCHEMBL12800994 0.72 TTR (0.35) TTRERN1ESR1HSP90AB1ESR2
SCHEMBL11898569 0.69 ERN1 (0.43) ERN1ESR1HSP90AB1ESR2NSD3
SCHEMBL1670808 0.67 TTR (0.34) TTRESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011042477-A1 SUBSTITUTED PYRROLES AND IMIDAZOLES AS ESTROGEN RECEPTOR LIGANDS KARO BIO AB (SE) 2011-04-14 WO disclosed
WO-2011042477-A1 SUBSTITUTED PYRROLES AND IMIDAZOLES AS ESTROGEN RECEPTOR LIGANDS KARO BIO AB (SE) 2011-04-14 WO disclosed