SCHEMBL16709352

SCHEMBL16709352

NC(=O)c1ccc2[nH]c3ccc(Br)cc3c2c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT1 Q96EB6 2/20 0.50
PARP1 P09874 1/20 0.50
CHUK O15111 1/20 0.46
HTR1B P28222 2/20 0.46
AR P10275 1/20 0.45
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
CYP1A2 P05177 2/20 0.44
HTR1A P08908 1/20 0.44
TSHR P16473 1/20 0.44
HTR1D P28221 1/20 0.44
HTR2C P28335 1/20 0.44
HTR7 P34969 1/20 0.44
HTR5A P47898 1/20 0.44
HTR6 P50406 1/20 0.44
HSD17B10 Q99714 1/20 0.44
PRNP P04156 1/20 0.44
CYP2C9 P11712 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15486127 0.84 MEN1 (0.56) SIRT1CHUKARMEN1KMT2A
SCHEMBL11810570 0.82 KIF11 (0.57) PARP1HTR1BMEN1KMT2ARAB9A
SCHEMBL1180875 0.81 KDM4E (0.59) MEN1KMT2ARAB9AHTR7HSD17B10
SCHEMBL29643250 0.81 KDM4E (0.59) MEN1KMT2ARAB9AHTR7HSD17B10
SCHEMBL16709582 0.79 KIF11 (0.62) PARP1HTR1BMEN1KMT2ANPC1
SCHEMBL25658280 0.79 HTR1B (0.46) PARP1HTR1BMEN1KMT2ARAB9A
SCHEMBL29366993 0.79 CHUK (0.64) CHUKARCYP1A2HSD17B10PRNP
SCHEMBL38602 0.79 CHUK (0.64) CHUKARCYP1A2HSD17B10PRNP
Hydrochloric Acid SCHEMBL8594443 0.78 KDM4E (0.56) MEN1KMT2ARAB9AHTR7HSD17B10
Hydrochloric Acid SCHEMBL8594438 0.78 KDM4E (0.56) MEN1KMT2ARAB9AHTR7HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9243281-B2 Neuroprotective chemicals and methods for identifying and using same BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2016-01-26 US disclosed
US-9243281-B2 Neuroprotective chemicals and methods for identifying and using same BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2016-01-26 US disclosed
US-20150132783-A1 Neuroprotective Chemicals and Methods for Identifying and Using Same UNIVERSITY OF IOWA RESEARCH FOUNDATION (US) 2015-05-14 US disclosed
US-20150132783-A1 Neuroprotective Chemicals and Methods for Identifying and Using Same UNIVERSITY OF IOWA RESEARCH FOUNDATION (US) 2015-05-14 US disclosed
WO-2015070237-A1 NEUROPROTECTIVE CHEMICALS AND METHODS FOR IDENTIFYING AND USING SAME BOARD OF REGENTS OF THE UNIVERSITY OF TEXAS SYSTEM (US) 2015-05-14 WO disclosed