SCHEMBL16713201

SCHEMBL16713201

O=C(CC[C@@H](C(=O)O)N(Cc1ccccc1)Cc1ccccc1)Cc1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
CES2 O00748 1/20 0.40
CES1 P23141 1/20 0.40
AKR1B1 P15121 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
EPOR P19235 2/20 0.40
CPA3 P15088 1/20 0.38
KMT2A Q03164 3/20 0.38
MEN1 O00255 2/20 0.38
REN P00797 1/20 0.38
VNN1 O95497 1/20 0.37
TRPM8 Q7Z2W7 1/20 0.37
CYP1A2 P05177 1/20 0.37
CNR2 P34972 1/20 0.37
CHRNB2 P17787 1/20 0.37
CHRNB4 P30926 1/20 0.37
CHRNA3 P32297 1/20 0.37
CHRNA4 P43681 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19384899 0.85 CPA3 (0.53) NPC1RAB9AEPORCPA3CYP1A2
SCHEMBL536547 0.85 CPA3 (0.53) NPC1RAB9AEPORCPA3CYP1A2
SCHEMBL536546 0.85 CPA3 (0.53) NPC1RAB9AEPORCPA3CYP1A2
Hydrochloric Acid SCHEMBL3025758 0.84 CPA3 (0.51) NPC1RAB9AEPORCPA3CYP1A2
Hydrochloric Acid SCHEMBL3025760 0.84 CPA3 (0.51) NPC1RAB9AEPORCPA3CYP1A2
SCHEMBL8398528 0.83 NPC1 (0.41) NPC1RAB9AEPORCPA3KMT2A
SCHEMBL840672 0.79 LMNA (0.46) L3MBTL1NPC1RAB9AEPORKMT2A
SCHEMBL841385 0.79 LMNA (0.46) L3MBTL1NPC1RAB9AEPORKMT2A
SCHEMBL842165 0.78 GRIK1 (0.53) TDP1NPC1RAB9AEPORKMT2A
SCHEMBL22444192 0.78 KMT2A (0.44) NPC1RAB9AEPORKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20150141615-A1 ALDEHYDE ACETAL BASED PROCESSES FOR THE MANUFACTURE OF MACROCYCLIC DEPSIPEPTIDES AND NEW INTERMEDIATES NOVARTIS AG (CH) 2015-05-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150141615-A1 ALDEHYDE ACETAL BASED PROCESSES FOR THE MANUFACTURE OF MACROCYCLIC DEPSIPEPTIDES AND NEW INTERMEDIATES DNPEP, VIP, ALDH16A1 TDP1 4092/4885L3MBTL1 2147/4885CES2 2186/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.