SCHEMBL167172

SCHEMBL167172

CS(=O)(=O)c1cccc(-c2ccc3ccsc3c2)c1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 4/20 0.46
LIMK1 P53667 1/20 0.45
CA12 O43570 2/20 0.43
CA2 P00918 2/20 0.43
NR1H2 P55055 5/20 0.41
NR1H3 Q13133 1/20 0.41
BCL9 O00512 1/20 0.41
CTNNB1 P35222 1/20 0.41
KCNH2 Q12809 2/20 0.40
LOXL2 Q9Y4K0 1/20 0.40
PIK3CD O00329 1/20 0.39
PIK3CG P48736 1/20 0.39
PIP4K2C Q8TBX8 2/20 0.39
SCD O00767 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL165069 0.88 CA2 (0.57) PTGS2LIMK1CA12CA2NR1H2
SCHEMBL6742234 0.82 PTGS2 (0.42) PTGS2CA12CA2
SCHEMBL6243674 0.78 KCNH2 (0.50) PTGS2LIMK1NR1H2NR1H3KCNH2
SCHEMBL145018 0.77 LIMK1 (0.44) PTGS2LIMK1NR1H2NR1H3KCNH2
SCHEMBL13742552 0.76 DYRK1A (0.48) CA12CA2
SCHEMBL13472079 0.75 CA12 (0.45) CA12CA2
SCHEMBL2140712 0.73 PTGS2 (0.53) PTGS2NR1H2NR1H3KCNH2LOXL2
SCHEMBL6737344 0.72 CA2 (0.51) PTGS2CA12CA2
SCHEMBL3712310 0.71 PI4KA (0.73) LIMK1PIK3CDPIK3CG
SCHEMBL28846692 0.71 SCD (0.54) PTGS2CA12CA2KCNH2LOXL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2611774-A1 DI-AZETIDINYL DIAMIDE AS MONOACYLGLYCEROL LIPASE INHIBITORS Janssen Pharmaceutica, N.V. (BE) 2013-07-10 EP claimed
WO-2012030907-A1 DI-AZETIDINYL DIAMIDE AS MONOACYLGLYCEROL LIPASE INHIBITORS JANSSEN PHARMACEUTICA NV (BE) 2012-03-08 WO claimed