SCHEMBL16720176

SCHEMBL16720176

c1ccn(-c2ccc3[nH]ccc3c2)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.47
AHR P35869 4/20 0.47
NR4A2 P43354 2/20 0.47
CYP2A6 P11509 2/20 0.47
F7 P08709 1/20 0.47
LTA4H P09960 1/20 0.47
F3 P13726 1/20 0.47
USP2 O75604 1/20 0.47
GAA P10253 1/20 0.47
ALOX15 P16050 1/20 0.47
RAD51 Q06609 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
TRPA1 O75762 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
ITGB2 P05107 1/20 0.43
ICAM1 P05362 1/20 0.43
ITGAL P20701 1/20 0.43
CA4 P22748 1/20 0.43
CA6 P23280 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16720407 0.85 AHR (0.47) NPC1AHRCYP2A6TRPA1CA1
SCHEMBL27417145 0.84 CYP2A6 (0.43) NPC1AHRNR4A2CYP2A6F7
SCHEMBL8404071 0.79 GABRP (0.48) NPC1AHRNR4A2CYP2A6F7
SCHEMBL9091484 0.78 CYP19A1 (0.57) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL803139 0.74 KMT2A (0.50) NPC1USP2CA1CA2MAPT
SCHEMBL26259748 0.74 MAPT (0.50) NPC1GAANPSR1MAPTCYP1A2
SCHEMBL26259867 0.72 CYP19A1 (0.48) NPC1GAANPSR1MAPTCYP1A2
SCHEMBL3340549 0.72 LTA4H (0.48) AHRNR4A2CYP2A6F7LTA4H
SCHEMBL1122665 0.72 GABRP (0.48) NPC1AHRNR4A2CYP2A6F7
SCHEMBL25203062 0.72 GABRP (0.45) NPC1AHRNR4A2CYP2A6F7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3068758-A1 EBNA1 INHIBITORS AND THEIR METHOD OF USE The Wistar Institute Of Anatomy And Biology (US) 2016-09-21 EP disclosed
WO-2015073864-A1 EBNA1 INHIBITORS AND THEIR METHOD OF USE THE WISAR INSTITUTE OF ANATOMY AND BIOLOGY (US) 2015-05-21 WO disclosed