SCHEMBL16728601

SCHEMBL16728601

CC(=O)Nc1ccc(C#N)c(Cl)c1

nearest known ligand 0.63

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.63
IDO1 P14902 1/20 0.59
LMNA P02545 1/20 0.53
GAA P10253 1/20 0.53
RORC P51449 3/20 0.51
AR P10275 4/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
BLM P54132 1/20 0.49
SLC22A12 Q96S37 3/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6816427 0.91 IDO1 (0.66) ALDH1A1IDO1LMNAGAA
SCHEMBL1192659 0.87 ALDH1A1 (0.63) ALDH1A1RORCSMN1; SMN2BLMSLC22A12
SCHEMBL307278 0.86 IDO1 (0.62) ALDH1A1IDO1LMNAGAAAR
SCHEMBL16722682 0.85 IDO1 (0.60) ALDH1A1IDO1LMNAGAARORC
SCHEMBL7234787 0.85 RORC (0.53) ALDH1A1RORCSMN1; SMN2
SCHEMBL202348 0.84 IDO1 (0.54) ALDH1A1IDO1LMNAGAARORC
SCHEMBL6816436 0.84 ALDH1A1 (0.48) ALDH1A1IDO1LMNAGAARORC
SCHEMBL8351343 0.84 ALDH1A1 (0.79) ALDH1A1LMNASMN1; SMN2
SCHEMBL12050119 0.81 AR (0.58) IDO1AR
SCHEMBL13909401 0.81 IDO1 (0.54) ALDH1A1IDO1LMNAGAARORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3147278-A1 COMPOUND FOR TREATING BREAST CANCER AND PROGESTIN-DEPENDENT CONDITIONS University of Tennessee Research Foundation (US) 2017-03-29 EP disclosed
WO-2015073767-A1 SUBSTITUTED 4,5,6,7-TETRAHYDROPYRAZOLO[1,5-A]PYRAZINE DERIVATIVES AS CASEIN KINASE 1 D/E INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2015-05-21 WO disclosed