SCHEMBL1672901

SCHEMBL1672901

Cn1cncc1-c1c(-c2ccc(O)cc2)c(Cl)n(C)c1C(N)=NO

nearest known ligand 0.36

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 3/20 0.36
LDLR P01130 1/20 0.31
PCSK9 Q8NBP7 1/20 0.31
HTR1A P08908 2/20 0.31
HTR7 P34969 2/20 0.31
HTR6 P50406 2/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
DRD2 P14416 1/20 0.31
HPGDS O60760 1/20 0.30
BRAF P15056 1/20 0.30
MAPK3 P27361 1/20 0.30
MAPK1 P28482 1/20 0.30
GSK3B P49841 1/20 0.30
DYRK1A Q13627 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1672900 0.80 IDO1 (0.36) IDO1LDLRPCSK9HPGDSGSK3B
SCHEMBL1672283 0.77 ESR1 (0.32)
SCHEMBL1672285 0.77 ESR1 (0.32)
SCHEMBL1670636 0.76 USP7 (0.30)
SCHEMBL1671213 0.76 NTRK1 (0.38) BRAFMAPK3MAPK1
SCHEMBL1670618 0.73
SCHEMBL1670617 0.73
SCHEMBL14676514 0.72 IDO1 (0.36) IDO1HTR1AHTR7HTR6CYP3A4
SCHEMBL14676515 0.72 IDO1 (0.36) IDO1HTR1AHTR7HTR6CYP3A4
SCHEMBL1671132 0.71 KDM1A (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011042477-A1 SUBSTITUTED PYRROLES AND IMIDAZOLES AS ESTROGEN RECEPTOR LIGANDS KARO BIO AB (SE) 2011-04-14 WO claimed