SCHEMBL1672900

SCHEMBL1672900

Cn1cncc1-c1c(-c2ccc(O)cc2)c(Cl)n(C)c1C(=N)NO

nearest known ligand 0.38

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 3/20 0.36
GSK3B P49841 3/20 0.32
DYRK1A Q13627 3/20 0.32
LDLR P01130 1/20 0.31
PCSK9 Q8NBP7 1/20 0.31
HPGDS O60760 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1672901 0.80 IDO1 (0.36) IDO1GSK3BDYRK1ALDLRPCSK9
SCHEMBL1670634 0.76 AKT1 (0.31)
SCHEMBL1672287 0.76 ESR1 (0.32)
SCHEMBL1671210 0.75 USP7 (0.30)
SCHEMBL21141726 0.73 IDO1 (0.36) IDO1GSK3BDYRK1AHPGDS
SCHEMBL1670619 0.73
SCHEMBL1671138 0.71 ESR1 (0.30)
SCHEMBL1670522 0.71 SENP1 (0.30)
SCHEMBL1670633 0.70 GSK3B (0.34) GSK3B
SCHEMBL1671012 0.70

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011042477-A1 SUBSTITUTED PYRROLES AND IMIDAZOLES AS ESTROGEN RECEPTOR LIGANDS KARO BIO AB (SE) 2011-04-14 WO claimed