SCHEMBL1672934

SCHEMBL1672934

COc1nc(Br)cnc1I

nearest known ligand 0.42

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CCR4 P51679 15/20 0.42
CCR5 P51681 1/20 0.38
EDNRA P25101 4/20 0.38
MAPK1 P28482 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL609085 0.80 CCR4 (0.45) CCR4CCR5EDNRA
SCHEMBL30416654 0.80 CCR4 (0.45) CCR4CCR5EDNRA
SCHEMBL20399659 0.77 CCR4 (0.35) CCR4EDNRA
SCHEMBL29364914 0.77 CCR4 (0.43) CCR4CCR5EDNRA
SCHEMBL14970085 0.77 CCR4 (0.43) CCR4CCR5EDNRA
SCHEMBL68083 0.77 CCR4 (0.43) CCR4CCR5EDNRA
SCHEMBL19785488 0.76 APP (0.50)
SCHEMBL30296090 0.76 APP (0.50)
SCHEMBL19193244 0.75 CCR4 (0.42) CCR4CCR5EDNRA
SCHEMBL31133084 0.75 CCR4 (0.42) CCR4CCR5EDNRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 58 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4709381-A1 PARP1 INHIBITOR COMPOUNDS Duke Street Bio Limited (GB) 2026-03-18 EP disclosed
US-20250270195-A1 PD-1/PD-L1 INHIBITORS GILEAD SCIENCES INC (US) 2025-08-28 US disclosed
US-12338233-B2 PD-1/Pd-L1 inhibitors GILEAD SCIENCES, INC. (US) 2025-06-24 US disclosed
WO-2025029075-A1 NOVEL BIPHENYL DERIVATIVE AS PD-L1 INHIBITOR (주)아이랩 2025-02-06 WO disclosed
EP-4499630-A1 BCL-XL INHIBITORS BeiGene, Ltd. (KY) 2025-02-05 EP disclosed
US-20250034128-A1 BCL-XL INHIBITORS BEIGENE, LTD. (KY) 2025-01-30 US disclosed
WO-2024256377-A1 PARP1 INHIBITOR COMPOUNDS Duke Street Bio Limited (GB) 2024-12-19 WO disclosed
CN-118974033-A Bcl-xL inhibitors 百济神州有限公司 2024-11-15 CN disclosed
US-20240336601-A1 4-PHENYL-INDOLE DERIVATIVES AND RELATED USES CHULALONG UNIVERSITY (TH) 2024-10-10 US disclosed
CN-118084940-A PD-1/PD-L1 inhibitors 吉利德科学公司 2024-05-28 CN disclosed
US-20160326143-A1 COMPOUNDS AND USES ASTRAZENECA AB (SE) 2016-11-10 US disclosed
WO-2016177845-A1 CYCLOPROPANE CARBOXYLIC ACID DERIVATIVES AND PHARMACEUTICAL USES THEREOF ASTRAZENECA AB (SE) 2016-11-10 WO disclosed
US-20160326143-A1 COMPOUNDS AND USES ASTRAZENECA AB (SE) 2016-11-10 US disclosed
US-20160326143-A1 COMPOUNDS AND USES ASTRAZENECA AB (SE) 2016-11-10 US disclosed
WO-2016177845-A1 CYCLOPROPANE CARBOXYLIC ACID DERIVATIVES AND PHARMACEUTICAL USES THEREOF ASTRAZENECA AB (SE) 2016-11-10 WO disclosed
EP-2491026-A1 NOVEL HETEROARYL IMIDAZOLES AND HETEROARYL TRIAZOLES AS GAMMA-SECRETASE MODULATORS Pfizer Inc. (US) 2012-08-29 EP disclosed
US-20120202787-A1 Novel Heteroaryl Imidazoles And Heteroaryl Triazoles As Gamma-Secretase Modulators PFIZER INC. 2012-08-09 US disclosed
US-20120202787-A1 Novel Heteroaryl Imidazoles And Heteroaryl Triazoles As Gamma-Secretase Modulators PFIZER INC. 2012-08-09 US disclosed
US-20120202787-A1 Novel Heteroaryl Imidazoles And Heteroaryl Triazoles As Gamma-Secretase Modulators PFIZER INC. 2012-08-09 US disclosed
WO-2011048525-A1 NOVEL HETEROARYL IMIDAZOLES AND HETEROARYL TRIAZOLES AS GAMMA-SECRETASE MODULATORS PFIZER INC. (US) 2011-04-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120202787-A1 Novel Heteroaryl Imidazoles And Heteroaryl Triazoles As Gamma-Secretase Modulators BACE1, BACE2, GSAP CCR4 4864/4885CCR5 3843/4885EDNRA 2997/4885
US-12338233-B2 PD-1/Pd-L1 inhibitors PDCD1, CD274, PDCD1LG2 CCR4 960/4885CCR5 403/4885EDNRA 2239/4885
US-20250034128-A1 BCL-XL INHIBITORS BCL2, BCL2L1, BCL2L10 CCR4 3798/4885CCR5 3066/4885EDNRA 4075/4885
US-20240336601-A1 4-PHENYL-INDOLE DERIVATIVES AND RELATED USES PDCD1, PDCD1LG2, CD274 CCR4 1229/4885CCR5 315/4885EDNRA 1063/4885
US-20250270195-A1 PD-1/PD-L1 INHIBITORS PDCD1, CD274, PDCD1LG2 CCR4 960/4885CCR5 403/4885EDNRA 2239/4885
US-20160326143-A1 COMPOUNDS AND USES LTC4S, LTB4R2, LTA4H CCR4 1098/4885CCR5 940/4885EDNRA 992/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.