SCHEMBL1673353

SCHEMBL1673353

Fc1ccc(CC2CCCN2)cc1

nearest known ligand 0.61

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.61
LTA4H P09960 1/20 0.49
PLG P00747 1/20 0.47
HTR2A P28223 1/20 0.46
HTR6 P50406 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10132251 1.00 POLB (0.61) POLBLTA4HPLGHTR2AHTR6
SCHEMBL23477699 0.93 POLB (0.67) POLBLTA4HPLGHTR2A
SCHEMBL29472327 0.86 PLG (0.50) POLBPLG
SCHEMBL23572347 0.84 PLG (0.47) POLBLTA4HPLG
SCHEMBL1990261 0.81 POLB (0.61) POLBLTA4HHTR6
SCHEMBL1443794 0.81 POLB (0.61) POLBLTA4HHTR6
SCHEMBL18577442 0.81 POLB (0.61) POLBLTA4HHTR6
SCHEMBL22456087 0.81 POLB (0.51) POLBHTR2AHTR6
SCHEMBL10132295 0.81 POLB (0.61) POLBLTA4HHTR6
SCHEMBL19654759 0.81 POLB (0.61) POLBLTA4HHTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4069366-B1 ATM KINASE INHIBITORS AND COMPOSITIONS AND METHODS OF USE THEREOF CHDI FOUNDATION INC (US) 2025-03-19 EP disclosed
US-11685734-B2 ATM kinase inhibitors and compositions and methods of use thereof CHDI FOUNDATION, INC. (US) 2023-06-27 US disclosed
US-20210188827-A1 ATM KINASE INHIBITORS AND COMPOSITIONS AND METHODS OF USE THEREOF CHDI FOUNDATION, INC. 2021-06-24 US disclosed
US-9650362-B2 Inhibitors PROBIODRUG AG (DE) 2017-05-16 US disclosed
US-20160039795-A1 NOVEL INHIBITORS VIVORYON THERAPEUTICS N.V. (DE) 2016-02-11 US disclosed
US-9173885-B2 Inhibitors PROBIODRUG AG (DE) 2015-11-03 US disclosed
US-20140065095-A1 NOVEL INHIBITORS VIVORYON THERAPEUTICS N.V. (DE) 2014-03-06 US disclosed
US-8486940-B2 Inhibitors PROBIODRUG AG (DE) 2013-07-16 US disclosed
US-8354413-B2 Quinolin-4-one and 4-oxodihydrocinnoline derivatives as inhibitors of poly(ADP-ribose) polymerase (PARP) Istituto di Ricerche di Biologia Molecolare P. Angeletti, S.R.L. (IT) 2013-01-15 US disclosed
CN-102695546-A Heterocylcic derivatives as inhibitors of glutaminyl cyclase PROBIODRUG AG 2012-09-26 CN disclosed
US-20110207720-A1 QUINOLIN-4-ONE AND 4-OXODIHYRDOCINNOLINE DERIVATIVES AS INHIBITORS OF POLY(ADP-RIBOSE) POLYMERASE (PARP) ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI S.R.L. (IT) 2011-08-25 US disclosed
US-20110092501-A1 NOVEL INHIBITORS PROBIODRUG AG (DE) 2011-04-21 US disclosed
EP-2193121-A1 QUINOLIN-4-ONE AND 4-OXODIHYDROCINNOLINE DERIVATIVES AS INHIBITORS OF POLY(ADP-RIBOSE)POLYMERASE (PARP) Istituto Di Ricerche Di Biologia Molecolare P. Angeletti S.P.A. (IT) 2010-06-09 EP disclosed
WO-2009027730-A1 QUINOLIN-4-ONE AND 4-OXODIHYDROCINNOLINE DERIVATIVES AS INHIBITORS OF POLY(ADP-RIBOSE)POLYMERASE (PARP) ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI S.P.A. (IT) 2009-03-05 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110092501-A1 NOVEL INHIBITORS GLUL, QPCT, GLS POLB 1125/4885LTA4H 2295/4885PLG 1338/4885
US-11685734-B2 ATM kinase inhibitors and compositions and methods of use thereof ATM, CHEK2, CHEK1 POLB 260/4885LTA4H 4678/4885PLG 3706/4885
US-20160039795-A1 NOVEL INHIBITORS GLUL, QPCT, GLS POLB 1125/4885LTA4H 2295/4885PLG 1338/4885
US-20110207720-A1 QUINOLIN-4-ONE AND 4-OXODIHYRDOCINNOLINE DERIVATIVES AS INHIBITORS OF POLY(ADP-RIBOSE) POLYMERASE (PARP) PARP1, PARP2, PARP11 POLB 25/4885LTA4H 3458/4885PLG 415/4885
US-20140065095-A1 NOVEL INHIBITORS GLUL, QPCT, GLS POLB 1125/4885LTA4H 2295/4885PLG 1338/4885
US-20210188827-A1 ATM KINASE INHIBITORS AND COMPOSITIONS AND METHODS OF USE THEREOF ATM, CHEK2, CHEK1 POLB 260/4885LTA4H 4678/4885PLG 3706/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.