SCHEMBL16740656

SCHEMBL16740656

COc1ccc(C=CC(=O)c2ccccc2OC)cc1OC

nearest known ligand 0.80

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 8/20 0.80
MAOB P27338 2/20 0.80
ACHE P22303 1/20 0.80
ABCB1 P08183 1/20 0.74
ABCC1 P33527 1/20 0.74
PDE4A P27815 1/20 0.72
PDE4B Q07343 1/20 0.72
PDE4C Q08493 1/20 0.72
PDE4D Q08499 1/20 0.72
SMN1; SMN2 Q16637 4/20 0.72
MEN1 O00255 3/20 0.72
KMT2A Q03164 3/20 0.72
MAPT P10636 2/20 0.72
PTGS1 P23219 1/20 0.67
PTGS2 P35354 1/20 0.67
CYP3A4 P08684 2/20 0.65
ALDH1A1 P00352 2/20 0.65
HPGD P15428 2/20 0.65
ALOX15 P16050 2/20 0.65
MAPK1 P28482 2/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16740655 1.00 ABCG2 (0.80) ABCG2MAOBACHEABCB1ABCC1
SCHEMBL17549125 0.90 MAPT (0.72) ABCG2MAOBACHEABCB1ABCC1
SCHEMBL2944203 0.89 ABCG2 (0.76) ABCG2MAOBACHEABCB1ABCC1
SCHEMBL25191764 0.89 ABCG2 (0.76) ABCG2MAOBACHEABCB1ABCC1
SCHEMBL2944206 0.89 ABCG2 (0.76) ABCG2MAOBACHEABCB1ABCC1
SCHEMBL25202039 0.89 ABCG2 (0.76) ABCG2MAOBACHEABCB1ABCC1
SCHEMBL25191295 0.89 PTGS1 (0.85) ABCG2MAOBACHEMEN1KMT2A
SCHEMBL25223438 0.89 MAOB (1.00) ABCG2MAOBACHEPDE4APDE4B
SCHEMBL634191 0.89 MAOB (1.00) ABCG2MAOBACHEPDE4APDE4B
SCHEMBL31233232 0.89 ABCG2 (0.76) ABCG2MAOBACHEABCB1ABCC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015075051-A1 ALLOSTERIC INHIBITORS OF ATYPICAL PROTEIN KINASES C UNIVERSITAET DES SAARLANDES (DE) 2015-05-28 WO disclosed