SCHEMBL16746751

SCHEMBL16746751

CC(c1ccc2ccccc2c1)c1cc(N)[nH]n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 3/20 0.47
ADRA2B P18089 3/20 0.47
ADRA2C P18825 3/20 0.47
UGT2B7 P16662 1/20 0.45
IKBKB O14920 1/20 0.39
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
AOC3 Q16853 2/20 0.37
CYP1A2 P05177 2/20 0.37
CYP2D6 P10635 1/20 0.37
TSHR P16473 1/20 0.37
HIF1A Q16665 1/20 0.37
ATM Q13315 1/20 0.36
MMP9 P14780 1/20 0.35
ALDH1A1 P00352 1/20 0.35
CYP3A4 P08684 1/20 0.35
HSD17B10 Q99714 1/20 0.35
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
HTR2B P41595 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16746780 0.82 KMT2A (0.41) MEN1KMT2ACYP1A2ALDH1A1HTR2C
SCHEMBL11642492 0.82 KMT2A (0.41) MEN1KMT2ACYP1A2ALDH1A1HTR2C
SCHEMBL16746783 0.80 JAK2 (0.41) MEN1KMT2ACYP1A2ALDH1A1CYP3A4
SCHEMBL16746749 0.78 JAK2 (0.39) MEN1KMT2ACYP1A2ALDH1A1
SCHEMBL16746779 0.77 PTGS1 (0.47) MEN1KMT2ACYP1A2CYP2D6ALDH1A1
SCHEMBL16746781 0.77 CYP3A4 (0.41) AOC3CYP1A2CYP2D6ALDH1A1CYP3A4
SCHEMBL16746820 0.76 DAO (0.40) ALDH1A1HTR2C
SCHEMBL16746862 0.76 ADRB2 (0.41) ADRA2AADRA2BADRA2CIKBKBMEN1
SCHEMBL16746857 0.76 IKBKB (0.39) IKBKBTSHRALDH1A1HSD17B10
SCHEMBL16746775 0.76 DHFR (0.40) AOC3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015076353-A1 3-ALKYLPYRAZOLOPYRIDINE DERIVATIVE 第一三共株式会社 2015-05-28 WO disclosed