SCHEMBL16758175

SCHEMBL16758175

CCC(F)(CC)CN1CCC(COc2ccc(-c3ccc(C(=O)NC(=O)[C@@H]4C[C@@H](O)CN4)cc3F)nc2)CC1

nearest known ligand 0.36

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP4F2 P78329 6/20 0.36
CYP4A11 Q02928 6/20 0.36
HPGDS O60760 4/20 0.35
GPR119 Q8TDV5 8/20 0.34
SCN9A Q15858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16757859 0.92 CYP4F2 (0.36) CYP4F2CYP4A11HPGDSGPR119SCN9A
SCHEMBL16758058 0.92 CYP4F2 (0.36) CYP4F2CYP4A11HPGDSGPR119SCN9A
SCHEMBL16757836 0.90 GPR119 (0.42) CYP4F2CYP4A11HPGDSGPR119
SCHEMBL16758005 0.87 WDR5 (0.37) HPGDS
SCHEMBL16757762 0.87 GPR119 (0.35) CYP4F2CYP4A11GPR119SCN9A
SCHEMBL16757750 0.86 GPR119 (0.46) CYP4F2CYP4A11HPGDSGPR119SCN9A
SCHEMBL16757851 0.85 CYP4F2 (0.36) CYP4F2CYP4A11HPGDSGPR119SCN9A
SCHEMBL16758261 0.83 GPR119 (0.38) CYP4F2CYP4A11HPGDSGPR119
SCHEMBL16757862 0.82 GPR119 (0.43) CYP4F2CYP4A11HPGDSGPR119
SCHEMBL16757902 0.82 SSTR5 (0.43) CYP4F2CYP4A11HPGDSGPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3074384-A1 AMIDE DERIVATIVES FOR GPR119 AGONIST Chong Kun Dang Pharmaceutical Corp. (KR) 2016-10-05 EP claimed
WO-2015080446-A1 AMIDE DERIVATIVES FOR GPR119 AGONIST CHONG KUN DANG PHARMACEUTICAL CORP. (KR) 2015-06-04 WO claimed
EP-3074384-A1 AMIDE DERIVATIVES FOR GPR119 AGONIST Chong Kun Dang Pharmaceutical Corp. (KR) 2016-10-05 EP disclosed
WO-2015080446-A1 AMIDE DERIVATIVES FOR GPR119 AGONIST CHONG KUN DANG PHARMACEUTICAL CORP. (KR) 2015-06-04 WO disclosed