SCHEMBL16759779

SCHEMBL16759779

Cn1cc(C(=O)OCC(F)(F)F)cc(Cl)c1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JMJD6 Q6NYC1 1/20 0.43
NPC1 O15118 5/20 0.40
RAB9A P51151 5/20 0.40
ALDH1A1 P00352 5/20 0.40
LMNA P02545 4/20 0.40
XBP1 P17861 3/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
NPSR1 Q6W5P4 3/20 0.40
CYP1A2 P05177 2/20 0.40
HSP90AA1 P07900 2/20 0.40
HPGD P15428 2/20 0.40
CYP2C19 P33261 2/20 0.40
MAPT P10636 3/20 0.39
HTT P42858 3/20 0.39
BAZ2B Q9UIF8 1/20 0.39
BAZ2A Q9UIF9 1/20 0.39
SLC6A3 Q01959 1/20 0.38
ATM Q13315 1/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23217732 0.77 CYP1A2 (0.46) ALDH1A1SMN1; SMN2CYP1A2CYP2C19MAPT
SCHEMBL6649202 0.76 KMT2A (0.49) ALDH1A1SMN1; SMN2NPSR1CYP1A2CYP2C19
SCHEMBL9248628 0.76 SLC6A3 (0.45) JMJD6NPC1RAB9AALDH1A1LMNA
SCHEMBL480184 0.72 TTR (0.45) RAB9ABAZ2BBAZ2AMEN1KMT2A
SCHEMBL9246003 0.71 SLC6A3 (0.41) JMJD6NPC1RAB9AXBP1SMN1; SMN2
SCHEMBL18045051 0.69 MEN1 (0.44) ALDH1A1LMNASMN1; SMN2CYP1A2CYP2C19
SCHEMBL19002423 0.69 KMT2A (0.43) NPC1RAB9AALDH1A1LMNACYP1A2
SCHEMBL27301733 0.68 BAZ2B (0.46) ALDH1A1LMNANPSR1CYP1A2HSP90AA1
SCHEMBL7558237 0.68 MAPT (0.49) JMJD6LMNASMN1; SMN2CYP1A2CYP2C19
SCHEMBL1496824 0.68 MAPK1 (0.55) JMJD6NPC1RAB9AALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3074400-A1 NEW OCTAHYDRO-CYCLOBUTA [1,2-c;3,4-c']DIPYRROL-2-YL F. Hoffmann-La Roche AG (CH) 2016-10-05 EP disclosed
WO-2015078803-A1 NEW OCTAHYDRO-CYCLOBUTA [1,2-c;3,4-c']DIPYRROL-2-YL F. HOFFMANN-LA ROCHE AG (CH) 2015-06-04 WO disclosed