SCHEMBL16770909

SCHEMBL16770909

Cn1c(-c2ccccc2)c(I)c2cncnc21

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 11/20 0.45
CYP3A4 P08684 7/20 0.45
TSHR P16473 4/20 0.45
CLK4 Q9HAZ1 2/20 0.45
LRRK2 Q5S007 1/20 0.40
GRM4 Q14833 1/20 0.39
HSD17B10 Q99714 6/20 0.37
CYP2C9 P11712 5/20 0.37
ALDH1A1 P00352 7/20 0.36
CYP2C19 P33261 4/20 0.36
ADORA3 P0DMS8 1/20 0.35
ADORA2A P29274 1/20 0.35
ADORA2B P29275 1/20 0.35
ADORA1 P30542 1/20 0.35
PI4KA P42356 1/20 0.35
PI4K2B Q8TCG2 1/20 0.35
PI4K2A Q9BTU6 1/20 0.35
PI4KB Q9UBF8 1/20 0.35
USP2 O75604 5/20 0.35
MAPK1 P28482 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4781863 0.78 FEN1 (0.42) TSHRLRRK2GRM4HSD17B10ALDH1A1
SCHEMBL14976832 0.77 TLR7 (0.41) CYP1A2CYP3A4TSHRCLK4LRRK2
SCHEMBL13172843 0.70 PI4KA (0.41) CYP1A2CYP3A4TSHRCLK4GRM4
SCHEMBL1609982 0.69 GPR3 (0.52) CYP1A2CYP3A4TSHRCLK4LMNA
SCHEMBL24828099 0.69 CYP1A2 (0.50) CYP1A2CYP3A4TSHRCLK4HSD17B10
SCHEMBL15170653 0.69 CYP1A2 (0.41) CYP1A2CYP3A4TSHRCLK4GRM4
SCHEMBL2628310 0.66 FEN1 (0.45) CYP1A2CYP3A4TSHRCLK4GRM4
SCHEMBL16771011 0.66 CCNB2 (0.51) CYP1A2CYP3A4TSHRCLK4HSD17B10
SCHEMBL9611672 0.66 CYP1A2 (0.65) CYP1A2CYP3A4TSHRCLK4HSD17B10
SCHEMBL2628313 0.65 CYP1A2 (0.34) CYP1A2CYP3A4TSHRCLK4GRM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015078417-A1 PYRROLOPYRIMIDINE COMPOUND AND USE THEREOF IN PREPARATION OF HYPOGLAECEMIC DRUG 四川好医生药业集团有限公司 2015-06-04 WO disclosed