SCHEMBL16775437

SCHEMBL16775437

CC(F)(F)c1cccc(-n2ccc(-c3ccc(C(=O)O)cc3)c2)c1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RXRA P19793 6/20 0.49
RXRB P28702 5/20 0.49
RXRG P48443 3/20 0.43
MEN1 O00255 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
KMT2A Q03164 1/20 0.41
SRD5A2 P31213 1/20 0.40
P2RY14 Q15391 1/20 0.39
ADH5 P11766 2/20 0.39
CFTR P13569 1/20 0.38
COMT P21964 1/20 0.38
NR1H4 Q96RI1 1/20 0.38
DHODH Q02127 2/20 0.38
NOTUM Q6P988 1/20 0.38
EGFR P00533 1/20 0.38
GRIN1 Q05586 1/20 0.37
GRIN2B Q13224 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL182393 0.90 RXRA (0.51) RXRARXRBRXRGMEN1NPC1
SCHEMBL16775447 0.89 MEN1 (0.50) RXRARXRBMEN1NPC1RAB9A
SCHEMBL16775446 0.83 RXRA (0.42) RXRARXRBRXRGP2RY14ADH5
SCHEMBL182269 0.82 RXRA (0.49) RXRARXRBRXRGMEN1KMT2A
SCHEMBL182330 0.81 TUBB4A (0.48) RXRARXRBRXRGMEN1KMT2A
SCHEMBL182600 0.81 BCL2L1 (0.47) ADH5COMTNOTUM
SCHEMBL2712103 0.81 AURKA (0.45) RXRARXRBRXRGADH5DHODH
SCHEMBL17125394 0.80 MEN1 (0.65) RXRARXRBRXRGMEN1NPC1
SCHEMBL2712235 0.79 KMT2A (0.58) RXRARXRBMEN1NPC1RAB9A
SCHEMBL2708139 0.79 TUBB4A (0.53) RXRARXRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9051342-B2 Pyrazole or triazole compounds and their use for the manufacture of a medicament for treating somatic mutation related diseases PTC THERAPEUTICS, INC. (US) 2015-06-09 US disclosed