SCHEMBL1678003

SCHEMBL1678003

O=C(O)C=CC(=O)c1cccc(Cl)c1Cl

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.60
ERCC5 P28715 1/20 0.49
FEN1 P39748 1/20 0.49
CXCL12 P48061 1/20 0.48
JAK2 O60674 1/20 0.45
ALDH1A1 P00352 4/20 0.44
P2RX7 Q99572 2/20 0.44
TAS1R3 Q7RTX0 1/20 0.41
TAS1R1 Q7RTX1 1/20 0.41
TAS1R2 Q8TE23 1/20 0.41
CES2 O00748 1/20 0.41
CES1 P23141 1/20 0.41
MAPT P10636 3/20 0.40
KMT2A Q03164 2/20 0.40
CYP2C9 P11712 1/20 0.40
HTT P42858 2/20 0.40
NPSR1 Q6W5P4 2/20 0.40
KDM4E B2RXH2 1/20 0.40
MEN1 O00255 1/20 0.40
POLB P06746 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10919848 0.85 ALDH1A1 (0.57) TSHRERCC5FEN1CXCL12ALDH1A1
SCHEMBL10919845 0.85 ALDH1A1 (0.57) TSHRERCC5FEN1CXCL12ALDH1A1
SCHEMBL11221211 0.82 ALDH1A1 (0.47) TSHRALDH1A1P2RX7CES2CES1
SCHEMBL11221208 0.82 ALDH1A1 (0.47) TSHRALDH1A1P2RX7CES2CES1
SCHEMBL27741821 0.81 MAPT (0.60) TSHRCXCL12ALDH1A1MAPTKMT2A
SCHEMBL8723935 0.79 TSHR (0.61) TSHRERCC5FEN1CXCL12JAK2
SCHEMBL5272752 0.76 TSHR (0.58) TSHRERCC5FEN1CXCL12JAK2
SCHEMBL5272753 0.76 TSHR (0.58) TSHRERCC5FEN1CXCL12JAK2
SCHEMBL97298 0.76 TSHR (1.00) TSHRERCC5FEN1JAK2ALDH1A1
SCHEMBL29904615 0.76 TSHR (1.00) TSHRERCC5FEN1JAK2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2308847-A1 Substituted pyridines as inhibitors of dipeptidyl peptidase IV and their application for the treatment of diabetes and related diseases EMC microcollections GmbH (DE) 2011-04-13 EP disclosed