SCHEMBL16794847

SCHEMBL16794847

COc1cccc(C(Br)C=O)c1F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 2/20 0.40
TLR2 O60603 1/20 0.38
TLR1 Q15399 1/20 0.38
TLR6 Q9Y2C9 1/20 0.38
CA1 P00915 4/20 0.37
CA2 P00918 4/20 0.37
ACHE P22303 2/20 0.37
HTT P42858 2/20 0.36
POLB P06746 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
CA12 O43570 2/20 0.34
CA7 P43166 2/20 0.34
CA9 Q16790 2/20 0.34
CA14 Q9ULX7 2/20 0.34
CA4 P22748 1/20 0.34
NFE2L2 Q16236 2/20 0.34
HDAC4 P56524 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL169082 0.84 CA1 (0.46) ERN1TLR2TLR1TLR6CA1
SCHEMBL3417280 0.80 ERN1 (0.40) ERN1HTTPOLBHTR2AHTR2C
SCHEMBL3415066 0.77 TLR2 (0.43) ERN1TLR2TLR1TLR6CA1
SCHEMBL20550915 0.77 CES2 (0.43) ERN1HDAC4
SCHEMBL5786635 0.77 KDM4E (0.38) ERN1HTTPOLBNFE2L2ALDH1A1
SCHEMBL8523806 0.76 POLB (0.43) ERN1TLR2TLR1TLR6CA1
SCHEMBL22827469 0.74 KRAS (0.44) ERN1CA1CA2ACHEHTT
SCHEMBL84457 0.74 LPAR1 (0.44) CA1CA2ACHEHTTPOLB
SCHEMBL16962349 0.72 CA1 (0.37) ERN1CA1CA2ACHEHTT
SCHEMBL23343773 0.72 CA1 (0.39) CA1CA2ACHEHTTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015088564-A1 P2X4 RECEPTOR MODULATING COMPOUNDS SUNOVION PHARMACEUTICALS INC. (US) 2015-06-18 WO disclosed
WO-2015088565-A1 P2X4 RECEPTOR MODULATING COMPOUNDS AND METHODS OF USE THEREOF SUNOVION PHARMACEUTICALS INC. (US) 2015-06-18 WO disclosed